SCHEMBL11277201

SCHEMBL11277201

COC1CSC2=C(SC1)C(OC(=O)N1CCN(C)CC1)N(c1ccc3ccc(Cl)cc3n1)C2=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.47
MAPT P10636 1/20 0.47
RECQL P46063 1/20 0.47
GABRA1 P14867 1/20 0.47
GABRA3 P34903 1/20 0.47
GABRA2 P47869 1/20 0.47
GABRB2 P47870 1/20 0.47
GABRA4 P48169 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
HRH4 Q9H3N8 8/20 0.36
HRH3 Q9Y5N1 5/20 0.35
HTR3A P46098 1/20 0.34
FNTA P49354 3/20 0.34
FNTB P49356 3/20 0.34
HRH1 P35367 1/20 0.34
ALOX15 P16050 1/20 0.32
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11836835 0.89 TSHR (0.48) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11266410 0.87 TSHR (0.63) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11263246 0.86 ADORA3 (0.44) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11262906 0.84 ADORA3 (0.42) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11266274 0.83 ADORA3 (0.40) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11264550 0.81 HRH3 (0.35) HRH4HRH3HTR3APDE10A
SCHEMBL11668941 0.80 MAPT (0.47) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL4729760 0.78 ADORA3 (0.75) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11267142 0.78 TSHR (0.51) ADORA3MAPTRECQLGABRA1GABRA3
SCHEMBL11268377 0.78 MAPT (0.35) ADORA3MAPTRECQLGABRA1GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4327095-A TRANQUICIZERS, ANTICONVULSANTS DECONTRACTURANTS AND HYPNOGENIC AGENTS RHONE-POULENC INDUSTRIES (FR) 1982-04-27 US claimed
US-4327095-A TRANQUICIZERS, ANTICONVULSANTS DECONTRACTURANTS AND HYPNOGENIC AGENTS RHONE-POULENC INDUSTRIES (FR) 1982-04-27 US disclosed