SCHEMBL1126845

SCHEMBL1126845

Cc1cc(C)nc(OCCOc2ccc(NC(=O)C(=O)c3c(-c4ccccc4)c(C)cn3C)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.41
HCRTR2 O43614 2/20 0.41
KCNA5 P22460 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36
MAPT P10636 3/20 0.35
RXFP1 Q9HBX9 1/20 0.35
CHRNA7 P36544 2/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
THRB P10828 1/20 0.34
PORCN Q9H237 2/20 0.34
ALDH1A1 P00352 1/20 0.34
DGAT1 O75907 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1126575 0.86 MCHR1 (0.36) KCNA5TDP1KMT2AMEN1NPC1
SCHEMBL1991373 0.84 HCRTR1 (0.39) HCRTR1HCRTR2KCNA5SMN1; SMN2TDP1
SCHEMBL1644580 0.82 MAPT (0.37) HCRTR1HCRTR2KCNA5SMN1; SMN2TDP1
SCHEMBL2231282 0.81 SMN1; SMN2 (0.41) HCRTR1HCRTR2KCNA5SMN1; SMN2TDP1
SCHEMBL1990047 0.80 HCRTR1 (0.38) HCRTR1HCRTR2KCNA5SMN1; SMN2TDP1
SCHEMBL1646398 0.80 SMN1; SMN2 (0.51) HCRTR1HCRTR2SMN1; SMN2TDP1KMT2A
SCHEMBL1646743 0.79 LMNA (0.40) HCRTR1HCRTR2KCNA5SMN1; SMN2KMT2A
SCHEMBL1646859 0.79 SMN1; SMN2 (0.38) HCRTR1HCRTR2KCNA5SMN1; SMN2TDP1
SCHEMBL2231172 0.79 LMNA (0.43) HCRTR1HCRTR2SMN1; SMN2TDP1TP53
SCHEMBL2233127 0.79 LMNA (0.40) HCRTR1HCRTR2KCNA5SMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed