SCHEMBL1126958

SCHEMBL1126958

CN(C)CCn1cc(-c2ccccc2)cc1C(=O)C(=O)Cl

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
CNR2 P34972 1/20 0.38
HTR6 P50406 8/20 0.37
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
GPR142 Q7Z601 1/20 0.36
UTS2R Q9UKP6 1/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR1D P28221 1/20 0.35
FAAH O00519 1/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1988726 0.78 CCNC (0.40) ALDH1A1CYP1A2CCNCCDK8CNR2
SCHEMBL1127844 0.76 KDM4E (0.41) ALDH1A1CYP1A2POLBCCNCCDK8
SCHEMBL1126509 0.74 HTR2A (0.42) HTR6HTR2AHTR2CHTR1D
SCHEMBL1126911 0.74 HTR2C (0.41) ALDH1A1CYP1A2POLBCNR2HTR6
SCHEMBL1126999 0.67 ESR1 (0.48) ALDH1A1CYP1A2POLBCCNCCDK8
SCHEMBL1127347 0.67 CNR1 (0.50) ALDH1A1CCNCCDK8CNR2USP2
SCHEMBL2834581 0.66 CCNC (0.43) ALDH1A1POLBCCNCCDK8KDM4E
SCHEMBL30740984 0.64 HTR2C (0.45) ALDH1A1CYP1A2POLBCNR2HTR6
SCHEMBL1126815 0.64 BRD4 (0.58) ALDH1A1POLBCCNCCDK8KDM4E
SCHEMBL1127225 0.63 CCNC (0.41) ALDH1A1CCNCCDK8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
EP-2626361-A1 Pyrrole antifungal agents F2G Limited (GB) 2013-08-14 EP disclosed
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed