SCHEMBL1126815

SCHEMBL1126815

Cn1cc(-c2ccccc2)cc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.58
CCNC P24863 1/20 0.51
CDK8 P49336 1/20 0.51
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
MCL1 Q07820 1/20 0.44
CYP2C9 P11712 2/20 0.44
LDHA P00338 2/20 0.44
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
BRD9 Q9H8M2 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KMO O15229 1/20 0.41
NR4A2 P43354 2/20 0.41
HDAC10 Q969S8 1/20 0.40
AR P10275 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12582221 0.85 CCNC (0.49) BRD4CCNCCDK8KDM4EALDH1A1
SCHEMBL16115664 0.84 CCNC (0.73) BRD4CCNCCDK8KDM4EALDH1A1
SCHEMBL25181069 0.83 KDM4E (0.52) BRD4CCNCCDK8KDM4EALDH1A1
SCHEMBL1254366 0.82 NR4A2 (0.54) BRD4CCNCCDK8KDM4EALDH1A1
SCHEMBL16691879 0.81 CCNC (0.45) BRD4CCNCCDK8MCL1CYP2C9
SCHEMBL16691871 0.80 KDM1A (0.51) BRD4CCNCCDK8KDM4EALDH1A1
SCHEMBL8461460 0.80 CYP2C9 (0.55) ALDH1A1GLACYP2C9KMT2AMEN1
SCHEMBL1126661 0.79 P2RY12 (0.51) BRD4KDM4EALDH1A1GAACYP2C9
SCHEMBL27660324 0.78 LDHA (0.41) BRD4KDM4EALDH1A1MCL1LDHA
SCHEMBL17266950 0.77 MAPT (0.45) BRD4CCNCCDK8KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250346575-A1 ISOINDOLINONE DERIVATIVE HAVING GLUTARIMIDE MOTHER NUCLEUS, AND USE THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2025-11-13 US disclosed
EP-4431505-A1 ISOINDOLINONE DERIVATIVE HAVING GLUTARIMIDE MOTHER NUCLEUS, AND USE THEREOF Korea Research Institute of Chemical Technology (KR) 2024-09-18 EP disclosed
CN-118234721-A Isoindolinone derivative with glutarimide mother nucleus and application thereof 韩国化学研究院 2024-06-21 CN disclosed
WO-2023085785-A1 ISOINDOLINONE DERIVATIVE HAVING GLUTARIMIDE MOTHER NUCLEUS, AND USE THEREOF 한국화학연구원 2023-05-19 WO disclosed
US-9452168-B2 Pyrrole antifungal agents F2G LTD (GB) 2016-09-27 US disclosed
US-20150238500-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-08-27 US disclosed
US-8993574-B2 Pyrrole antifungal agents F2G LTD (GB) 2015-03-31 US disclosed
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
CN-103833775-A SIRTUIN MODULATING COMPOUNDS SIRTRIS PHARMACEUTICALS INC 2014-06-04 CN disclosed
WO-2010118208-A1 BENZOXAZEPIN-4- (5H) -YL DERIVATIVES AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-10-14 WO disclosed
WO-2010118208-A1 BENZOXAZEPIN-4- (5H) -YL DERIVATIVES AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-10-14 WO disclosed
CN-101801981-A Sirtuin-modulating thiazolopyridine compounds SIRTRIS PHARMACEUTICALS INC 2010-08-11 CN disclosed
EP-2170905-A2 SIRTUIN MODULATING THIAZOLOPYRIDINE COMPOUNDS Sirtris Pharmaceuticals, Inc. (US) 2010-04-07 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed
US-20090105246-A1 Sirtuin modulating compounds SIRTRIS PHARMACEUTICALS, INC. (US) 2009-04-23 US disclosed
US-20090105246-A1 Sirtuin modulating compounds SIRTRIS PHARMACEUTICALS, INC. (US) 2009-04-23 US disclosed
US-20090105246-A1 Sirtuin modulating compounds SIRTRIS PHARMACEUTICALS, INC. (US) 2009-04-23 US disclosed
WO-2008156869-A2 SIRTUIN MODULATING THIAZOLOPYRIDINE COMPOUNDS SIRTRIS PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed
WO-2008156869-A2 SIRTUIN MODULATING THIAZOLOPYRIDINE COMPOUNDS SIRTRIS PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090105246-A1 Sirtuin modulating compounds SIRT1, SIRT3, SIRT2 BRD4 156/4885CCNC 3260/4885CDK8 796/4885
US-20150238500-A1 PYRROLE ANTIFUNGAL AGENTS FOXM1, PYCR1, ARG1 BRD4 3630/4885CCNC 2243/4885CDK8 3349/4885
US-20250346575-A1 ISOINDOLINONE DERIVATIVE HAVING GLUTARIMIDE MOTHER NUCLEUS, AND USE THEREOF CRBN, IDH1, IDH2 BRD4 324/4885CCNC 2659/4885CDK8 1117/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.