SCHEMBL1126966

SCHEMBL1126966

CCOC(=O)c1c(-c2ccccc2)c(C(=O)OCC)n(C)c1C(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.53
MAPT P10636 7/20 0.52
ALDH1A1 P00352 6/20 0.52
KDM4E B2RXH2 5/20 0.52
HPGD P15428 4/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
GAA P10253 4/20 0.52
LMNA P02545 3/20 0.52
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
TDP1 Q9NUW8 1/20 0.48
GRM6 O15303 1/20 0.47
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
TP53 P04637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127045 0.84 TSHR (0.68) TSHRMAPTALDH1A1KDM4EHPGD
SCHEMBL1126660 0.83 MAPT (0.46) TSHRMAPTALDH1A1KDM4EHPGD
SCHEMBL1127080 0.82 TSHR (0.55) TSHRMAPTALDH1A1KDM4EHPGD
SCHEMBL1126962 0.80 TSHR (0.53) TSHRMAPTALDH1A1KDM4EHPGD
SCHEMBL21484965 0.77 TSHR (0.55) TSHRMAPTALDH1A1KDM4EHPGD
SCHEMBL1991365 0.77 TSHR (0.50) TSHRMAPTALDH1A1KDM4EHPGD
SCHEMBL1126774 0.76 GRIA4 (0.46) ALDH1A1KDM4ESMN1; SMN2LMNATDP1
SCHEMBL1127099 0.75 TSHR (0.57) TSHRMAPTALDH1A1KDM4EHPGD
SCHEMBL28645817 0.75 TSHR (0.54) TSHRMAPTALDH1A1KDM4EHPGD
SCHEMBL1126753 0.75 TSHR (0.53) TSHRMAPTALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
EP-2626361-A1 Pyrrole antifungal agents F2G Limited (GB) 2013-08-14 EP disclosed
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed