SCHEMBL28645817

SCHEMBL28645817

CCOC(=O)c1c(-c2ccccc2)c(C(=O)C(=O)OC)c(C)n1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.54
MAPT P10636 6/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
RAB9A P51151 3/20 0.50
NPC1 O15118 2/20 0.50
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 6/20 0.47
GAA P10253 5/20 0.47
HPGD P15428 3/20 0.47
LMNA P02545 2/20 0.47
KDM4E B2RXH2 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
USP2 O75604 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
MAPK1 P28482 1/20 0.43
AR P10275 2/20 0.43
GRM6 O15303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127045 0.87 TSHR (0.68) TSHRMAPTSMN1; SMN2RAB9ANPC1
SCHEMBL21484965 0.80 TSHR (0.55) TSHRMAPTSMN1; SMN2RAB9ANPC1
SCHEMBL1126753 0.78 TSHR (0.53) TSHRMAPTSMN1; SMN2RAB9ANPC1
SCHEMBL1127080 0.77 TSHR (0.55) TSHRMAPTSMN1; SMN2RAB9ANPC1
SCHEMBL1126743 0.76 AR (0.49) TSHRMAPTSMN1; SMN2RAB9ANPC1
SCHEMBL1126962 0.75 TSHR (0.53) TSHRMAPTSMN1; SMN2RAB9ANPC1
SCHEMBL1126966 0.75 TSHR (0.53) TSHRMAPTSMN1; SMN2RAB9ANPC1
SCHEMBL1991365 0.75 TSHR (0.50) TSHRMAPTSMN1; SMN2RAB9ANPC1
SCHEMBL1127099 0.73 TSHR (0.57) TSHRMAPTSMN1; SMN2RAB9ANPC1
SCHEMBL1126643 0.73 TSHR (0.54) TSHRMAPTSMN1; SMN2RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429396-A Five-membered heteroaromatic ring derivative and preparation method and application thereof 深圳市祥根生物医药有限公司 2021-09-24 CN disclosed