SCHEMBL11270002

SCHEMBL11270002

CCc1cc(F)cc(Br)c1NC(=O)NC(=N)N

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 4/20 0.38
CACNA1C Q13936 3/20 0.38
ALDH1A1 P00352 3/20 0.37
GAA P10253 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
KMT2A Q03164 2/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
DRD2 P14416 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2B P41595 1/20 0.32
IDH1 O75874 1/20 0.32
PKM P14618 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056054 0.90 SCN5A (0.46) SCN5ACACNA1CALDH1A1GAAKMT2A
SCHEMBL11268006 0.86 SCN5A (0.41) SCN5ACACNA1CALDH1A1CA12CA1
SCHEMBL11141127 0.85 GAA (0.49) ALDH1A1GAAKMT2AMAPTSMN1; SMN2
SCHEMBL11414104 0.85 SCN5A (0.39) SCN5ACACNA1CALDH1A1GAAKMT2A
SCHEMBL11265596 0.84 SCN5A (0.38) SCN5ACACNA1CKMT2AMAPTSMN1; SMN2
SCHEMBL11278876 0.84 SCN5A (0.38) SCN5ACACNA1CALDH1A1CA1CA2
SCHEMBL11053535 0.83 DRD2 (0.39) ALDH1A1GAACA12CA1CA2
SCHEMBL11431492 0.83 ALDH1A1 (0.52) ALDH1A1GAACA12CA1CA2
SCHEMBL11057583 0.81 SCN5A (0.46) SCN5ACACNA1CALDH1A1KMT2AMAPT
SCHEMBL10941132 0.78 CACNA1C (0.56) SCN5ACACNA1CALDH1A1DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed