SCHEMBL11270574

SCHEMBL11270574

COc1ccc(CCC2(Cn3ccnc3)SCCS2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
MAPT P10636 3/20 0.47
TDP1 Q9NUW8 3/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
ALDH1A1 P00352 2/20 0.47
TP53 P04637 2/20 0.47
CYP1A2 P05177 2/20 0.47
TSHR P16473 2/20 0.47
CYP2C9 P11712 2/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TRPM8 Q7Z2W7 1/20 0.47
CYP19A1 P11511 2/20 0.46
ORAI1 Q96D31 1/20 0.46
CYP2D6 P10635 1/20 0.45
NFKB1 P19838 1/20 0.45
CYP2C19 P33261 1/20 0.45
MTOR P42345 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11262523 0.95 CYP3A4 (0.45) CYP3A4MAPTTDP1MEN1KMT2A
SCHEMBL11254606 0.93 CYP3A4 (0.50) CYP3A4MAPTTDP1MEN1KMT2A
SCHEMBL11266898 0.89 CYP3A4 (0.49) CYP3A4MAPTTDP1MEN1KMT2A
SCHEMBL11259195 0.89 CYP3A4 (0.48) CYP3A4MAPTTDP1MEN1KMT2A
SCHEMBL11257564 0.88 KDM4E (0.50) ALDH1A1HMOX1LMNA
SCHEMBL11266913 0.88 HMOX1 (0.42) CYP3A4MAPTTDP1MEN1KMT2A
SCHEMBL11258574 0.88 CYP19A1 (0.48) CYP3A4MAPTTDP1MEN1KMT2A
SCHEMBL11261572 0.87 CYP3A4 (0.42) CYP3A4MAPTTDP1MEN1KMT2A
SCHEMBL11265311 0.86 HMOX1 (0.47) HMOX1
SCHEMBL10247104 0.86 CYP19A1 (0.51) CYP19A1HMOX1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4359475-A SPERMICIDES, MICROBIOCIDES OR ANTICONVULSANTS SYNTEX (U.S.A.) INC. (US) 1982-11-16 US claimed
US-4359475-A SPERMICIDES, MICROBIOCIDES OR ANTICONVULSANTS SYNTEX (U.S.A.) INC. (US) 1982-11-16 US disclosed