SCHEMBL11270978

SCHEMBL11270978

CCC(C)OC(=O)C(CCCc1cccc(C(F)(F)F)c1)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
CYP3A4 P08684 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
USP2 O75604 2/20 0.43
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
HTR2B P41595 2/20 0.43
NR1I2 O75469 1/20 0.43
ADRB1 P08588 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11242316 0.97 HDAC1 (0.46) HDAC1HDAC8CYP3A4CYP1A2CYP2D6
SCHEMBL11203787 0.86 MAPK1 (0.49) HDAC1HDAC8CYP3A4CYP1A2CYP2D6
SCHEMBL11360753 0.83 HDAC1 (0.56) HDAC1HDAC8CYP3A4CYP1A2CYP2D6
SCHEMBL11264972 0.83 ALDH1A1 (0.42) PPARGPPARAFFAR4MEN1KMT2A
SCHEMBL11293581 0.83 PPARG (0.52) TSHRPPARGPPARAKDM4E
SCHEMBL7236478 0.82 MTNR1A (0.49) HDAC1TSHRCHRM3
SCHEMBL11203309 0.81 MAPK1 (0.54) HDAC1HDAC8TSHREPHX1FFAR4
SCHEMBL11261128 0.80 MAPT (0.46) KMT2A
SCHEMBL11268642 0.78 MAPT (0.45)
SCHEMBL11261409 0.78 MAPT (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4324796-A HYPOGLYCEMIC AGENTS, HYPOKETONEMIC AGENTS BYK GULDEN LOMBERG CHEMISCHE FABRIK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1982-04-13 US disclosed