SCHEMBL11274435

SCHEMBL11274435

Cn1nc(-c2ccccc2)c2c(=O)[nH]c(N)nc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 7/20 0.55
PARP1 P09874 2/20 0.48
KDM4E B2RXH2 2/20 0.48
GRM5 P41594 1/20 0.48
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
CASP1 P29466 1/20 0.44
BRCA1 P38398 1/20 0.44
HTT P42858 1/20 0.44
CASP7 P55210 1/20 0.44
KMT2A Q03164 1/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PIK3CA P42336 2/20 0.44
MTOR P42345 1/20 0.44
RICTOR Q6R327 1/20 0.44
RPTOR Q8N122 1/20 0.44
MAPKAP1 Q9BPZ7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11277238 0.85 PIK3CG (0.55) XDHPIK3CAMTORRICTORRPTOR
SCHEMBL5237936 0.84 POLB (0.54) PARP1KDM4EGRM5MEN1MAPT
SCHEMBL5234610 0.83 PARP1 (0.50) PARP1KDM4EGRM5MEN1MAPT
SCHEMBL5233091 0.78 TNKS (0.50) PARP1KDM4EGRM5MAPTHSD17B10
SCHEMBL409487 0.77 PIK3CD (0.51) PARP1KDM4EGRM5MEN1MAPT
SCHEMBL11271238 0.77 DHFR (0.51) PARP1KDM4EPIK3CAMTORRICTOR
SCHEMBL5232552 0.77 HTT (0.53) PARP1KDM4EGRM5MAPTHTT
SCHEMBL5231510 0.75 PDE7A (0.64) HTT
SCHEMBL5231538 0.75 PDE5A (0.57) KDM4EHTTFGFR1FGFR2
SCHEMBL5230247 0.75 POLB (0.44) PARP1KDM4EGRM5HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4315932-A AND SULFANILAMIDES BURROUGHS WELLCOME CO. (US) 1982-02-16 US disclosed
US-4288365-A 1H-PYRIMIDO(4,5-C)-1,2-DIAZEPINES BURROUGHS WELLCOME CO. (US) 1981-09-08 US disclosed
US-4237289-A MICROBIOCIDES BURROUGHS WELLCOME CO. (US) 1980-12-02 US disclosed