SCHEMBL11271238

SCHEMBL11271238

COc1cc(-c2nn(C)c3nc(N)[nH]c(=O)c23)cc(OC)c1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.51
KDR P35968 3/20 0.43
PIK3CA P42336 2/20 0.43
MTOR P42345 2/20 0.43
PIK3CD O00329 1/20 0.43
ABL1 P00519 1/20 0.43
EGFR P00533 1/20 0.43
HCK P08631 1/20 0.43
SRC P12931 1/20 0.43
PIK3CB P42338 1/20 0.43
PIK3CG P48736 1/20 0.43
EPHB4 P54760 1/20 0.43
PRKDC P78527 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
PDE7A Q13946 1/20 0.42
PDGFRB P09619 10/20 0.40
RICTOR Q6R327 1/20 0.40
RPTOR Q8N122 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11274435 0.77 XDH (0.55) DHFRKDRPIK3CAMTORPIK3CD
SCHEMBL11401818 0.76 DHFR (0.40) DHFRHSP90AA1HSP90AB1PDE7AKDM4E
SCHEMBL11277238 0.74 PIK3CG (0.55) KDRPIK3CAMTORPIK3CDABL1
SCHEMBL4222317 0.70 TLR7 (0.47) DHFRKDRPIK3CAMTORPIK3CD
SCHEMBL11261653 0.69 PDE5A (0.46) PARP1
SCHEMBL5231538 0.68 PDE5A (0.57) PDE7AKDM4E
SCHEMBL28234764 0.67 PIK3CD (0.42) KDRPIK3CAMTORPIK3CDABL1
SCHEMBL11401227 0.67 BRD4 (0.37) DHFRMTORHSP90AA1HSP90AB1PDE7A
SCHEMBL11233557 0.67 PDE5A (0.40) PARP1
SCHEMBL28233679 0.66 MAPT (0.56) KDRPIK3CAMTORPIK3CDABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4315932-A AND SULFANILAMIDES BURROUGHS WELLCOME CO. (US) 1982-02-16 US disclosed
US-4288365-A 1H-PYRIMIDO(4,5-C)-1,2-DIAZEPINES BURROUGHS WELLCOME CO. (US) 1981-09-08 US disclosed
US-4237289-A MICROBIOCIDES BURROUGHS WELLCOME CO. (US) 1980-12-02 US disclosed