SCHEMBL11277547

SCHEMBL11277547

c1ccc2c(c1)cn1[nH]cnc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F12 P00748 1/20 0.34
PLAU P00749 1/20 0.34
NCF1 P14598 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
BACE1 P56817 1/20 0.34
ALDH1A1 P00352 6/20 0.34
HSD17B10 Q99714 3/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 2/20 0.31
GPR3 P46089 1/20 0.31
PDPK1 O15530 1/20 0.31
CYP2A6 P11509 2/20 0.31
TSHR P16473 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
RAB9A P51151 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
PARP1 P09874 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11212810 0.61 ALDH1A1 (0.46) ALDH1A1HSD17B10HPGDKDM4ETSHR
SCHEMBL11171017 0.56 ALDH1A1 (0.41) F12PLAUNCF1NOS3NOS1
SCHEMBL22721038 0.54 ALDH1A1 (0.55) ALDH1A1HSD17B10HPGDCYP2A6TSHR
Naphthalene SCHEMBL7097704 0.52 CYP2A6 (0.89) ALDH1A1HSD17B10HPGDCYP2A6TSHR
Phenanthrene SCHEMBL29477074 0.51 CYP2A6 (1.00) ALDH1A1HSD17B10HPGDCYP2A6TSHR
Phenanthrene SCHEMBL30932938 0.51 CYP2A6 (1.00) ALDH1A1HSD17B10HPGDCYP2A6TSHR
Phenanthrene SCHEMBL29358486 0.51 CYP2A6 (1.00) ALDH1A1HSD17B10HPGDCYP2A6TSHR
SCHEMBL4377802 0.51 ALDH1A1 (0.85) ALDH1A1HSD17B10HPGDCYP2A6TSHR
Phenanthrene SCHEMBL7643 0.51 CYP2A6 (1.00) ALDH1A1HSD17B10HPGDCYP2A6TSHR
Phenanthrene SCHEMBL27458043 0.51 CYP2A6 (1.00) ALDH1A1HSD17B10HPGDCYP2A6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4313950-A Antireproductive tricyclic ortho-fused nitrogen containing compounds GRUPPO LEPETIT S.P.A. (IT) 1982-02-02 US disclosed
US-4275066-A 1,2,4-TRIAZOLO(5.1A)ISOINDOZE, TRIAZOLO(5.1A) ISOQUINOLINE OR 1,2,4,-TRIAZOLO (5.1A)(2) BENZAZEPINE CONTRACEPTIVES GRUPPO LEPETIT S.P.A. (IT) 1981-06-23 US disclosed
US-4007276-A ANTIFERTILITY, ANTIINFLAMMATORY, ANALGESIC, CNS DEPRESSANT, MICROBIOCIDES GRUPPO LEPETIT, S.P.A. (IT) 1977-02-08 US disclosed