SCHEMBL11277754

SCHEMBL11277754

COc1cccc(C)c1NC(=N)NC(=N)N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.47
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
TAAR1 Q96RJ0 1/20 0.39
PKM P14618 2/20 0.39
S1PR2 O95136 1/20 0.38
S1PR4 O95977 1/20 0.38
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38
S1PR5 Q9H228 1/20 0.38
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2B P41595 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6695373 0.88 ATM (0.51) ATMCYP1A2CYP3A4CYP2C19TAAR1
SCHEMBL1740895 0.85 DRD2 (0.49) ATMCYP1A2CYP3A4CYP2C19PKM
SCHEMBL10939799 0.85 ATM (0.62) ATMCYP1A2CYP3A4CYP2C19PKM
SCHEMBL11142783 0.85 ATM (0.45) ATMCYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL11264335 0.85 ATM (0.47) ATMCYP1A2CYP3A4CYP2C19TAAR1
SCHEMBL11659758 0.84 KLK1 (0.39) ATMPKMDRD2HTR2AHTR2B
SCHEMBL11659085 0.81 CACNA1C (0.42) ALDH1A1KMT2AL3MBTL1KLK1KLK5
SCHEMBL11660887 0.78 DRD2 (0.40) PKMDRD2HTR2AHTR2BGRIN2D
SCHEMBL11842943 0.78 DRD2 (0.40) ATMCYP1A2CYP2C19PKMDRD2
SCHEMBL11665157 0.78 DRD2 (0.40) CYP1A2CYP2C19PKMDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4117165-A ANTIULCER, HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-09-26 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed