SCHEMBL11264335

SCHEMBL11264335

CNC(=N)NC(=N)Nc1c(C)cccc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.47
TAAR1 Q96RJ0 1/20 0.39
PKM P14618 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C19 P33261 2/20 0.38
S1PR2 O95136 1/20 0.38
S1PR4 O95977 1/20 0.38
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38
S1PR5 Q9H228 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
KMT2A Q03164 5/20 0.36
DRD4 P21917 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KCNK3 O14649 1/20 0.36
POLB P06746 1/20 0.36
KCNK9 Q9NPC2 1/20 0.36
PDE4A P27815 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10614877 0.87 ATM (0.60) ATMPKMCYP1A2CYP3A4CYP2C19
SCHEMBL11287194 0.85 POLB (0.42) ATMPKMCYP1A2CYP3A4CYP2C19
SCHEMBL11277754 0.85 ATM (0.47) ATMTAAR1PKMCYP1A2CYP3A4
SCHEMBL11267001 0.84 NLRP3 (0.37) ATMKMT2AL3MBTL1ALDH1A1GAA
SCHEMBL6695373 0.82 ATM (0.51) ATMTAAR1PKMCYP1A2CYP3A4
SCHEMBL11284491 0.81 CACNA1C (0.39) KMT2APOLBALDH1A1MEN1
SCHEMBL11277149 0.78 GAA (0.50) S1PR2S1PR4KMT2AALDH1A1MEN1
SCHEMBL11252206 0.78 ATM (0.50) ATMPKMCYP1A2CYP3A4CYP2C19
SCHEMBL11284346 0.78 POLB (0.47) ATMPKMCYP1A2CYP3A4CYP2C19
SCHEMBL11251266 0.76 ALDH1A1 (0.44) ATMPKMCYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed