SCHEMBL11278490

SCHEMBL11278490

O=c1nc2ccccc2nc2ncncc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.46
PDE5A O76074 1/20 0.39
KDM4E B2RXH2 2/20 0.37
GPR3 P46089 1/20 0.37
PLAUR Q03405 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
MAPT P10636 3/20 0.34
ALDH1A1 P00352 6/20 0.34
HSD17B10 Q99714 3/20 0.34
HPGD P15428 2/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
CYP1A2 P05177 5/20 0.34
CYP2C9 P11712 4/20 0.34
CYP3A4 P08684 3/20 0.34
TSHR P16473 2/20 0.34
CLK4 Q9HAZ1 1/20 0.34
CYP2C19 P33261 3/20 0.33
MAPK1 P28482 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22589760 0.83 PLAUR (0.47) EGFRKDM4EGPR3PLAURALDH1A1
SCHEMBL30124132 0.75 EGFR (0.54) EGFRKDM4EGPR3PIK3CDPIK3CA
SCHEMBL35632 0.75 EGFR (0.54) EGFRKDM4EGPR3PIK3CDPIK3CA
SCHEMBL8967704 0.74 CYP3A4 (0.46) KDM4EGPR3PLAURMAPTALDH1A1
SCHEMBL30362637 0.74 ACHE (0.57) EGFRKDM4EMAPTALDH1A1HSD17B10
SCHEMBL28614688 0.74 ACHE (0.57) EGFRKDM4EMAPTALDH1A1HSD17B10
SCHEMBL10916482 0.72 ESR1 (0.47) EGFRKDM4EMAPTALDH1A1HSD17B10
SCHEMBL23649973 0.69 EGFR (0.52) EGFRKDM4EGPR3PIK3CDPIK3CA
SCHEMBL15796997 0.69 KDM4E (0.65) EGFRPDE5AKDM4EMAPTALDH1A1
SCHEMBL18099789 0.68 KDM4E (0.50) EGFRPDE5AKDM4EGPR3PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4311700-A ANTIULCER, GASTROINTESTINAL DISORDERS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1982-01-19 US disclosed
EP-0024582-A1 Benzodiazepinones, process for their preparation and pharmaceutical compositions containing them Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1981-03-11 EP disclosed
WO-1981000568-A1 BENZODIAZEPINONES,A PROCESS FOR THEIR PREPARATION,THEIR USE AND MEDICAMENTS CONTAINING THEM BYK GULDEN LOMBERG CHEM FAB (DE) 1981-03-05 WO disclosed