SCHEMBL11279397

SCHEMBL11279397

Nc1ccc(Cl)nc1C(=O)c1ccccc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
MAPT P10636 1/20 0.43
ALOX15 P16050 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
CDK5 Q00535 3/20 0.39
CDK5R1 Q15078 3/20 0.39
RECQL P46063 1/20 0.39
CDK2 P24941 1/20 0.37
GSK3B P49841 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
ELANE P08246 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GAA P10253 2/20 0.37
POLB P06746 1/20 0.36
PKM P14618 2/20 0.36
FADS1 O60427 1/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11272310 0.84 RECQL (0.55) ALDH1A1CES2CES1RECQLGAA
SCHEMBL11716248 0.84 ALDH1A1 (0.46) ALDH1A1MAPTALOX15CES2CES1
SCHEMBL11714368 0.83 ALDH1A1 (0.44) ALDH1A1MAPTRECQLSMN1; SMN2GAA
SCHEMBL11717520 0.82 RECQL (0.37) ALDH1A1RECQLGAAPOLBMEN1
SCHEMBL11715323 0.82 MAPK13 (0.42) ALDH1A1MAPTALOX15RECQLELANE
SCHEMBL11712393 0.82 MAPK13 (0.43) ALDH1A1ALOX15RECQLELANENPC1
SCHEMBL11716112 0.81 CNR2 (0.51) CDK2GAANPC1LMNA
SCHEMBL28014540 0.80 ALDH1A1 (0.42) ALDH1A1MAPTALOX15CES2CES1
SCHEMBL3837048 0.80 ALDH1A1 (0.49) ALDH1A1MAPTALOX15CES2CES1
SCHEMBL11273463 0.78 GAA (0.44) ALDH1A1MAPTALOX15CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE31071-E 6-Aza-3H-1,4-benzodiazepines DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DE) 1982-11-02 US disclosed
US-4012397-A 2-Benzoyl-3-amino-pyridines DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DT) 1977-03-15 US disclosed
US-4008223-A SPASMOLYTIC, ANTIPHLOGISTIC, TRANQUILIZER DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DT) 1977-02-15 US disclosed
US-3969361-A 2-Benzoyl-3-amino-pyridines DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DT) 1976-07-13 US disclosed