SCHEMBL11280776

SCHEMBL11280776

CC1=C(OC(=O)OCCC#N)C(c2cccc(Cl)c2)C(OC(=O)OC(C)C)=C(C)N1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 12/20 0.44
CACNA1F O60840 2/20 0.40
CACNA1D Q01668 2/20 0.40
CACNA1S Q13698 2/20 0.40
CACNA1C Q13936 2/20 0.40
MEN1 O00255 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 2/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
THPO P40225 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11291917 0.90 CACNA1F (0.52) CACNA1FCACNA1DCACNA1SCACNA1CMEN1
SCHEMBL11500635 0.87 CACNA1B (0.46) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL10913858 0.85 MEN1 (0.57) CACNA1FCACNA1DCACNA1SCACNA1CMEN1
SCHEMBL11106245 0.83 CACNA1B (0.60) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL11281855 0.83 KDM4E (0.44) CACNA1BMEN1KMT2ATSHRMAPT
SCHEMBL10913259 0.81 CACNA1C (0.55) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL11005887 0.79 CACNA1B (0.49) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL11500155 0.79 ALDH1A1 (0.44) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL11276232 0.79 TSHR (0.39) CACNA1FCACNA1DCACNA1SCACNA1CCYP1A2
SCHEMBL11498937 0.79 POLB (0.44) MEN1KMT2ALMNATSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0011706-B1 PROCESS FOR THE PREPARATION OF DERIVATIVES OF 1,4-DIHYDROPYRIDINE-3-CARBOXYLIC ACID, DERIVATIVES OF 1,4-DIHYDROPYRIDINE-3-CARBOXYLIC ACID AND THE USE OF THESE DERIVATIVES FOR THE PREPARATION OF 1,4-DIHYDROPYRIDINE-3,5-DICARBOXYLATES BAYER AG (DE) 1982-03-03 EP disclosed
EP-0011706-A1 Process for the preparation of derivatives of 1,4-dihydropyridine-3-carboxylic acid, derivatives of 1,4-dihydropyridine-3-carboxylic acid and the use of these derivatives for the preparation of 1,4-dihydropyridine-3,5-dicarboxylates BAYER AG (DE) 1980-06-11 EP disclosed