SCHEMBL11283149

SCHEMBL11283149

CCOC(=O)C=C(N)c1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.49
ALDH1A1 P00352 3/20 0.48
POLB P06746 1/20 0.48
NPSR1 Q6W5P4 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
MAPT P10636 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
ADORA1 P30542 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
THRB P10828 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11283146 1.00 CES2 (0.49) CES2ALDH1A1POLBNPSR1TAS1R3
SCHEMBL3269421 0.86 NPSR1 (0.52) CES2ALDH1A1POLBNPSR1TAS1R3
SCHEMBL23124814 0.84 NQO2 (0.49) CES2ALDH1A1POLBNPSR1TAS1R3
SCHEMBL23124816 0.84 NQO2 (0.49) CES2ALDH1A1POLBNPSR1TAS1R3
SCHEMBL11386442 0.83 NPSR1 (0.50) CES2ALDH1A1NPSR1MAPTMEN1
SCHEMBL11386447 0.83 NPSR1 (0.50) CES2ALDH1A1NPSR1MAPTMEN1
SCHEMBL29779353 0.83 NPSR1 (0.50) CES2ALDH1A1NPSR1MAPTMEN1
SCHEMBL20028184 0.82 LMNA (0.51) CES2ALDH1A1POLBNPSR1MAPT
SCHEMBL11393110 0.82 PARP1 (0.53) ALDH1A1TAS1R3TAS1R1MAPTHTT
SCHEMBL11393086 0.82 PARP1 (0.53) ALDH1A1TAS1R3TAS1R1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4336389-A 2-Substituted-4-aryl-5-thiazolecarboxylic acids and their derivatives as safening agents MONSANTO COMPANY (US) 1982-06-22 US disclosed
US-4261728-A PREEMERGENT ACTIVITY MONSANTO COMPANY (US) 1981-04-14 US disclosed
US-4187099-A 3-Aryl-4-isothiazolecarboxylic acid and 3-aryl-4-isoxazolecarboxylic acid derivatives and their use as herbicides MONSANTO COMPANY (US) 1980-02-05 US disclosed
US-4144047-A SOYBEANS MONSANTO COMPANY (US) 1979-03-13 US disclosed