SCHEMBL11286152

SCHEMBL11286152

CCCn1c(=O)c2[nH]c(C)nc2n(CC(C)O)c1=O

nearest known ligand 0.77

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.59
PDE1A P54750 1/20 0.59
PDE1B Q01064 1/20 0.59
PDE1C Q14123 1/20 0.59
SIRT1 Q96EB6 1/20 0.54
SIRT3 Q9NTG7 1/20 0.54
SIRT5 Q9NXA8 1/20 0.54
ADORA1 P30542 1/20 0.51
ADORA2A P29274 1/20 0.51
ADORA2B P29275 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9430566 0.96 PDE2A (0.56) PDE2APDE1APDE1BPDE1CSIRT1
SCHEMBL10855561 0.90 PDE2A (0.73) PDE2APDE1APDE1BPDE1CSIRT1
SCHEMBL1063544 0.88 SIRT1 (0.68) SIRT1SIRT3SIRT5ADORA1ADORA2A
SCHEMBL9429916 0.83 PDE2A (0.53) PDE2APDE1APDE1BPDE1CSIRT1
SCHEMBL10859893 0.82 SIRT1 (0.61) SIRT1SIRT3SIRT5ADORA1ADORA2A
SCHEMBL10856971 0.82 SIRT1 (0.61) SIRT1SIRT3SIRT5ADORA1ADORA2A
SCHEMBL9430619 0.82 ADORA2A (0.61) SIRT1SIRT3SIRT5ADORA1ADORA2A
SCHEMBL4623475 0.81 PDE1A (0.71) PDE2APDE1APDE1BPDE1CSIRT1
SCHEMBL9430131 0.81 ADORA2A (0.56) SIRT1SIRT3SIRT5ADORA1ADORA2A
SCHEMBL9430769 0.80 ADORA2A (0.55) SIRT1SIRT3SIRT5ADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0001735-B1 XANTHINE DERIVATIVES HAVING ANTIALLERGIC ACTIVITY AND PHARMACOLOGICAL PREPARATIONS CONTAINING THEM Aktiebolaget DRACO (SE) 1982-09-01 EP disclosed