SCHEMBL9430769

SCHEMBL9430769

CCCn1c(=O)n(CCCCCO)c(=O)c2[nH]c(C)nc21

nearest known ligand 0.77

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.55
ADORA2B P29275 2/20 0.55
PDE4A P27815 1/20 0.55
PDE4B Q07343 1/20 0.55
PDE4C Q08493 1/20 0.55
PDE4D Q08499 1/20 0.55
SIRT1 Q96EB6 1/20 0.54
SIRT3 Q9NTG7 1/20 0.54
SIRT5 Q9NXA8 1/20 0.54
ADORA1 P30542 6/20 0.53
MEN1 O00255 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9430131 0.99 ADORA2A (0.56) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL9430619 0.95 ADORA2A (0.61) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL10856971 0.88 SIRT1 (0.61) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL10859893 0.88 SIRT1 (0.61) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL1063544 0.88 SIRT1 (0.68) ADORA2AADORA2BSIRT1SIRT3SIRT5
SCHEMBL9430349 0.85 PDE1A (0.67) ADORA2AADORA2BSIRT1SIRT3SIRT5
SCHEMBL7918903 0.85 ADORA1 (0.57) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL18834910 0.81 PDE2A (0.53) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL11066305 0.81 SIRT1 (0.54) ADORA2AADORA2BSIRT1SIRT3SIRT5
SCHEMBL9430688 0.81 PDE1A (0.68) ADORA2AADORA2BPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269841-B1 1-HYDROXYALKYL XANTHINES, PROCESSES FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM SOCIETE DES PRODUITS NESTLE S.A. (CH) 1992-11-11 EP claimed
EP-0269841-A1 1-Hydroxyalkyl xanthines, processes for their preparation and medicaments containing them SOCIETE DES PRODUITS NESTLE S.A. (CH) 1988-06-08 EP claimed
US-5338741-A Cardiotonic agents NESTEC S.A. (CH) 1994-08-16 US disclosed
EP-0269841-B1 1-HYDROXYALKYL XANTHINES, PROCESSES FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM SOCIETE DES PRODUITS NESTLE S.A. (CH) 1992-11-11 EP disclosed
US-5053433-A Photodiesterase inhibitor SOCIETE ANONYME DITE: L'OREAL (FR) 1991-10-01 US disclosed
EP-0269841-A1 1-Hydroxyalkyl xanthines, processes for their preparation and medicaments containing them SOCIETE DES PRODUITS NESTLE S.A. (CH) 1988-06-08 EP disclosed