SCHEMBL11287141

SCHEMBL11287141

O=C(Cc1nc(=O)[nH]cc1Br)c1cccs1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
LMNA P02545 4/20 0.44
ALDH1A1 P00352 3/20 0.44
POLB P06746 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GSK3B P49841 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.40
CTNNB1 P35222 3/20 0.40
WNT3A P56704 2/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HPGD P15428 4/20 0.39
ERCC5 P28715 1/20 0.39
FEN1 P39748 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11293448 0.84 GSK3B (0.45) NPC1RAB9ALMNAALDH1A1POLB
SCHEMBL11290653 0.84 ALDH1A1 (0.44) NPC1RAB9ALMNAALDH1A1POLB
SCHEMBL11285972 0.76 GRIN2D (0.37) NPC1RAB9APOLBMEN1KMT2A
SCHEMBL11347681 0.75 PARP1 (0.43) NPC1RAB9ALMNAPOLBKMT2A
SCHEMBL11292813 0.74 ALDH1A1 (0.49) NPC1RAB9ALMNAALDH1A1POLB
SCHEMBL17595406 0.65 ALDH1A1 (0.50) NPC1RAB9ALMNAALDH1A1POLB
SCHEMBL11586017 0.65 ALDH1A1 (0.50) NPC1RAB9ALMNAALDH1A1POLB
SCHEMBL17596624 0.65 NPC1 (0.43) NPC1RAB9ALMNAALDH1A1POLB
SCHEMBL9049816 0.65 RAB9A (0.64) NPC1RAB9ALMNAALDH1A1POLB
SCHEMBL18437367 0.64 ALDH1A1 (0.58) NPC1RAB9ALMNAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0044705-A1 Substituted pyrimidin-2-ones, the salts thereof, processes for their preparation, pharmaceutical compositions containing them and a method therefor GLAXO GROUP LIMITED (GB) 1982-01-27 EP disclosed