Ethylenediamine

Ethylenediamine

SCHEMBL11289433

COC(=O)c1c(Br)c(Br)c(Br)c(Br)c1C(=O)OC.NCCN

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3PDE3APDE3BPDE4APDE4BPDE4CPDE4D

The experimentally established mechanism targets of Ethylenediamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
PTPN1 P18031 1/20 0.39
LOXL2 Q9Y4K0 2/20 0.38
F2 P00734 1/20 0.37
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37
PRSS3 P35030 1/20 0.37
ALDH1A1 P00352 2/20 0.36
PRKCZ Q05513 1/20 0.36
MAPT P10636 3/20 0.35
KDM4E B2RXH2 4/20 0.35
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
TSHR P16473 2/20 0.34
KMT2A Q03164 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11572303 0.92 KDM4E (0.37) CA12CA1CA2CA7CA9
SCHEMBL11290085 0.90 PAOX (0.38) CA12CA1CA2CA7CA9
SCHEMBL5698060 0.89 CA12 (0.46) CA12CA1CA2CA7CA9
SCHEMBL31306912 0.89 CA12 (0.46) CA12CA1CA2CA7CA9
SCHEMBL11569953 0.84 ALDH1A1 (0.37) CA12CA1CA2CA7CA9
SCHEMBL8380519 0.81 CA1 (0.48) CA12CA1CA2CA7CA9
SCHEMBL9717113 0.80 F2 (0.45) CA12CA1CA2CA7CA9
SCHEMBL29049264 0.76 CA12 (0.48) CA12CA1CA2CA7CA9
Ethylenediamine SCHEMBL11297757 0.74 F2 (0.35) F2PRSS1PRSS2PRSS3ALDH1A1
Ethylenediamine SCHEMBL11627367 0.72 F2 (0.42) PTPN1F2PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4328357-A Process for preparing nitrogen compounds SAYTECH, INC. (US) 1982-05-04 US disclosed
US-4140862-A Salts of diamines and tetrahalophthalates CITIES SERVICE COMPANY (US) 1979-02-20 US disclosed