Ethylenediamine

Ethylenediamine

SCHEMBL11297757

NCCN.O=C(O)c1c(Br)c(Br)c(Br)c(Br)c1C(=O)OCCOC(=O)c1c(Br)c(Br)c(Br)c(Br)c1C(=O)O

nearest known ligand 0.35

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Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3PDE3APDE3BPDE4APDE4BPDE4CPDE4D

The experimentally established mechanism targets of Ethylenediamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
F2 P00734 3/20 0.35
PRSS1 P07477 3/20 0.35
PRSS2 P07478 3/20 0.35
PRSS3 P35030 3/20 0.35
SERPINE1 P05121 2/20 0.33
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
ALDH1A1 P00352 1/20 0.30
TP53 P04637 1/20 0.30
GLA P06280 1/20 0.30
CYP3A4 P08684 1/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HIF1A Q16665 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7783160 0.94 F2 (0.34) F2PRSS1PRSS2PRSS3SERPINE1
SCHEMBL27457725 0.86 TDP1 (0.38) F2PRSS1PRSS2PRSS3SERPINE1
Ethylenediamine SCHEMBL11627367 0.85 F2 (0.42) F2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL4456791 0.85 ALDH1A1 (0.33) F2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL29445809 0.84
SCHEMBL11871467 0.80 ESR1 (0.50) NPC1RAB9AALDH1A1TP53CYP3A4
SCHEMBL10717061 0.80 THRB (0.45) F2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL9157297 0.78 ALDH1A1 (0.47) NPC1RAB9AALDH1A1CYP3A4HPGD
SCHEMBL8470318 0.78 ALDH1A1 (0.49) NPC1RAB9AALDH1A1TP53CYP3A4
SCHEMBL7946728 0.78 ALDH1A1 (0.49) NPC1RAB9AALDH1A1TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4328357-A Process for preparing nitrogen compounds SAYTECH, INC. (US) 1982-05-04 US disclosed
US-4140862-A Salts of diamines and tetrahalophthalates CITIES SERVICE COMPANY (US) 1979-02-20 US disclosed