SCHEMBL112925

SCHEMBL112925

O=C(O)NCC(C(=O)Nc1ccc2cnccc2c1)c1ccc(OCC(=O)c2ccccc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 0.64
ROCK1 Q13464 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2775038 0.89 ROCK2 (0.57) ROCK2ROCK1
SCHEMBL9883133 0.89 ROCK2 (0.77) ROCK2ROCK1
Hydrochloric Acid SCHEMBL110782 0.88 ROCK2 (0.75) ROCK2ROCK1
SCHEMBL114093 0.86 ROCK2 (0.61) ROCK2ROCK1
SCHEMBL113081 0.83 ROCK2 (0.74) ROCK2ROCK1
SCHEMBL28631002 0.82 ROCK2 (0.75) ROCK2ROCK1
SCHEMBL16056711 0.82 ROCK2 (0.75) ROCK2ROCK1
SCHEMBL21774951 0.81 ROCK2 (0.76) ROCK2ROCK1
SCHEMBL115008 0.81 ROCK2 (0.76) ROCK2ROCK1
SCHEMBL111744 0.81 ROCK2 (0.60) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424842-A2 DUAL MECHANISM INHIBITORS FOR THE TREATMENT OF DISEASE Aerie Pharmaceuticals, Inc. (US) 2012-03-07 EP disclosed
EP-2424857-A1 DUAL-ACTION INHIBITORS AND METHODS OF USING SAME Aerie Pharmaceuticals, Inc. (US) 2012-03-07 EP disclosed
WO-2010127329-A1 DUAL-ACTION INHIBITORS AND METHODS OF USING SAME AERIE PHARMACEUTICALS, INC. (US) 2010-11-04 WO disclosed
WO-2010127330-A1 DUAL-ACTION INHIBITORS AND METHODS OF USING SAME AERIE PHAMACEUTICALS, INC. (US) 2010-11-04 WO disclosed
WO-2010126626-A2 DUAL MECHANISM INHIBITORS FOR THE TREATMENT OF DISEASE AERIE PHARMACEUTICALS, INC. (US) 2010-11-04 WO disclosed