SCHEMBL11293296

SCHEMBL11293296

Nc1cc(-c2ccccn2)n[nH]c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.54
BTK Q06187 1/20 0.47
PRMT5 O14744 2/20 0.47
WDR77 Q9BQA1 1/20 0.47
KDM4E B2RXH2 5/20 0.47
LMNA P02545 4/20 0.47
CCR1 P32246 3/20 0.47
CCR5 P51681 3/20 0.47
CCR8 P51685 3/20 0.47
CYP1A2 P05177 1/20 0.47
POLB P06746 1/20 0.47
METAP1 P53582 1/20 0.47
BLM P54132 1/20 0.47
HIF1A Q16665 1/20 0.47
DOHH Q9BU89 1/20 0.47
P4HTM Q9NXG6 1/20 0.47
PDE2A O00408 1/20 0.45
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
METAP2 P50579 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1593197 0.82 PIN1 (0.56) PIN1BTKKDM4ELMNACCR1
SCHEMBL30040683 0.82 PIN1 (0.56) PIN1BTKKDM4ELMNACCR1
SCHEMBL23202619 0.80 PIN1 (0.54) PIN1BTKPRMT5WDR77KDM4E
SCHEMBL31096555 0.80 PIN1 (0.54) PIN1BTKPRMT5WDR77KDM4E
SCHEMBL27598057 0.79 PIN1 (0.56) PIN1BTKPRMT5WDR77KDM4E
SCHEMBL1392639 0.77 ADORA3 (0.56) KDM4ECYP1A2POLBPDE2APDE3B
SCHEMBL4855164 0.76 PIN1 (0.66) PIN1BTKPRMT5WDR77KDM4E
SCHEMBL11245576 0.75 PRMT5 (0.49) PRMT5WDR77KDM4ELMNACYP1A2
SCHEMBL1528433 0.73 PIN1 (0.57) PIN1BTKKDM4ELMNACCR1
SCHEMBL9598073 0.73 BTK (0.50) PIN1BTKPRMT5WDR77KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4346221-A Preparation of 4-amino-6-(pyridinyl)-3(2H)-pyridazinones from 6-(pyridinyl)-3(2H)-pyridazinones STERLING DRUG INC. (US) 1982-08-24 US disclosed
US-4305943-A 4-Amino-6-(pyridinyl)-3(2H)-pyridazinones and their use as cardiotonics STERLING DRUG INC. (US) 1981-12-15 US disclosed