SCHEMBL11296183

SCHEMBL11296183

O=C1N=C(c2ccc(O)cc2)C(=O)N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.40
ESR1 P03372 3/20 0.39
ESR2 Q92731 1/20 0.39
SENP1 Q9P0U3 1/20 0.38
TDP2 O95551 1/20 0.38
RAB9A P51151 2/20 0.37
MEN1 O00255 2/20 0.37
MAPT P10636 2/20 0.37
KMT2A Q03164 2/20 0.37
NPC1 O15118 1/20 0.37
USP2 O75604 1/20 0.37
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TNKS O95271 2/20 0.37
PARP1 P09874 2/20 0.37
TNKS2 Q9H2K2 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1624199 0.80 ALDH1A1 (0.46) PTGS2TDP2MAPTKMT2AHPGD
SCHEMBL8093099 0.66 RARB (0.44)
SCHEMBL16492050 0.64 PTGS2 (0.52) PTGS2ESR1ESR2SENP1TDP2
SCHEMBL6551950 0.63
SCHEMBL6702892 0.63 PTGS2 (0.59) PTGS2ESR1ESR2SENP1TDP2
SCHEMBL6292004 0.60 ESR1 (1.00) ESR1ESR2RAB9AMEN1MAPT
SCHEMBL9090705 0.60 ESR1 (1.00) ESR1ESR2RAB9AMEN1MAPT
Hydroquinone SCHEMBL5712110 0.60 ESR1 (1.00) ESR1ESR2RAB9AMEN1MAPT
SCHEMBL30826784 0.60 ESR1 (1.00) ESR1ESR2RAB9AMEN1MAPT
SCHEMBL15632 0.60 ESR1 (1.00) ESR1ESR2RAB9AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0022492-B1 STEREO SELECTIVE RESOLUTION OF PHENYLGLYCINE DERIVATIVES WITH ENZYMERESINS BAYER AG (DE) 1982-09-29 EP disclosed
EP-0022492-A1 Stereo selective resolution of phenylglycine derivatives with enzymeresins BAYER AG (DE) 1981-01-21 EP disclosed
EP-0003786-B1 STEREOSELECTIVE SEPARATION OF PHENYLGLYCINE DERIVATIVES AND 4-HYDROXYPHENYLGLYCINE DERIVATIVES WITH ENZYME-CONTAINING POLYMERS BAYER AG (DE) 1980-12-10 EP disclosed