SCHEMBL11299409

SCHEMBL11299409

Cc1cc(N)ccc1N1CCN(C(C)(C)C)CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.65
ALDH1A1 P00352 8/20 0.65
GAA P10253 4/20 0.65
MEN1 O00255 3/20 0.65
THRB P10828 3/20 0.65
KMT2A Q03164 3/20 0.65
NR4A1 P22736 1/20 0.65
PTK2B Q14289 1/20 0.65
GFER P55789 3/20 0.60
RAD52 P43351 2/20 0.60
KDM4E B2RXH2 3/20 0.47
LMNA P02545 2/20 0.47
ALOX15 P16050 2/20 0.47
POLB P06746 1/20 0.41
HTT P42858 2/20 0.41
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A3 P47895 2/20 0.38
HSD17B10 Q99714 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15358737 0.88 MAPT (0.81) MAPTALDH1A1GAAMEN1THRB
SCHEMBL11296569 0.83 MAPT (0.66) MAPTALDH1A1GAAMEN1THRB
SCHEMBL6272228 0.82 ALDH1A1 (0.86) MAPTALDH1A1GAAMEN1THRB
SCHEMBL11364687 0.82 MAPT (0.60) MAPTALDH1A1GAAMEN1THRB
SCHEMBL25091069 0.81 MAPT (0.71) MAPTALDH1A1GAAMEN1THRB
Hydrochloric Acid SCHEMBL7051020 0.81 ALDH1A1 (0.89) MAPTALDH1A1GAAMEN1THRB
SCHEMBL187881 0.81 ALDH1A1 (0.71) MAPTALDH1A1GAAMEN1THRB
SCHEMBL29477783 0.81 ALDH1A1 (0.71) MAPTALDH1A1GAAMEN1THRB
SCHEMBL6156455 0.80 ALDH1A1 (0.96) MAPTALDH1A1GAAMEN1THRB
SCHEMBL7031588 0.80 ALDH1A1 (0.89) MAPTALDH1A1GAAMEN1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3694509-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Nuvation Bio Inc. (US) 2020-08-19 EP disclosed
WO-2019074981-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF GiraFpharma LLC (US) 2019-04-18 WO disclosed
EP-3083625-A1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS Almac Discovery Limited (GB) 2016-10-26 EP disclosed
WO-2015092431-A1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2015-06-25 WO disclosed
EP-2681221-A1 TRICYCLIC INHIBITORS OF KINASES AbbVie Inc. (US) 2014-01-08 EP disclosed
EP-2665724-A1 BICYCLIC INHIBITORS OF ALK AbbVie Inc. (US) 2013-11-27 EP disclosed
WO-2012161812-A1 TRICYCLIC INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2012-11-29 WO disclosed
WO-2012097682-A1 BICYCLIC INHIBITORS OF ALK ABBOTT LABORATORIES (US) 2012-07-26 WO disclosed