SCHEMBL11312445

SCHEMBL11312445

CCc1nc(-c2ccccc2)nc(N)c1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.57
RAB9A P51151 3/20 0.57
TP53 P04637 2/20 0.57
HSD17B10 Q99714 1/20 0.57
KMT2A Q03164 3/20 0.56
FABP3 P05413 1/20 0.47
FABP4 P15090 1/20 0.47
FABP5 Q01469 1/20 0.47
NPC1 O15118 2/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MAPT P10636 1/20 0.46
DHFR P00374 4/20 0.45
HEXA P06865 1/20 0.45
HEXB P07686 1/20 0.45
TSHR P16473 1/20 0.44
PDE4B Q07343 2/20 0.44
PDE4D Q08499 2/20 0.44
GAA P10253 1/20 0.43
ADORA3 P0DMS8 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5509874 0.83 KDM4E (0.55) KDM4ERAB9ATP53HSD17B10KMT2A
SCHEMBL31556277 0.75 DHFR (0.47) TP53KMT2AALDH1A1SMN1; SMN2DHFR
SCHEMBL11494053 0.74 KDM4E (0.73) KDM4ERAB9ATP53HSD17B10KMT2A
SCHEMBL27633592 0.74 KDM4E (0.54) KDM4ERAB9ATP53HSD17B10KMT2A
SCHEMBL5521948 0.72 KDM4E (0.56) KDM4ERAB9ATP53HSD17B10KMT2A
SCHEMBL5659586 0.72 GABRP (0.41) KDM4ERAB9ATP53HSD17B10KMT2A
SCHEMBL11908452 0.72 GABRP (0.41) KDM4ERAB9ATP53HSD17B10KMT2A
SCHEMBL5961069 0.72 FABP3 (0.49) KDM4ERAB9ATP53HSD17B10KMT2A
SCHEMBL3258197 0.72 TSHR (0.80) KDM4ERAB9ATP53HSD17B10KMT2A
SCHEMBL10377332 0.71 CFTR (0.47) RAB9ATP53KMT2ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4301281-A 7,8-Dihydro-2,5,8-trisubstituted-7-oxo-pyrido[2,3-d]-pyrimidine-6-carboxylic acid amides AMERICAN HOME PRODUCTS CORPORATION (US) 1981-11-17 US disclosed