SCHEMBL11319

SCHEMBL11319

CN(c1ccccc1)S(=O)(=O)c1ccccc1-c1ccc2cc(C(=O)O)n(O)c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 3/20 0.55
DAO P14920 1/20 0.45
KDM4E B2RXH2 3/20 0.40
PKM P14618 1/20 0.39
MCOLN3 Q8TDD5 1/20 0.38
MAPT P10636 2/20 0.36
HTT P42858 2/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MCL1 Q07820 1/20 0.36
LMNA P02545 1/20 0.36
PGR P06401 1/20 0.36
POLB P06746 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP1A2 P05177 1/20 0.35
ALOX12 P18054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14118492 0.84 LDHA (0.64) LDHADAOKDM4EMAPTHTT
SCHEMBL11316 0.82 LDHA (0.56) LDHADAOMAPTHTTSMN1; SMN2
SCHEMBL14118470 0.75 LDHA (0.56) LDHADAOMAPTHTTSMN1; SMN2
SCHEMBL14118481 0.73 LDHA (0.64) LDHADAOKDM4EMAPTHTT
SCHEMBL14118407 0.73 MAPT (0.51) LDHADAOMCOLN3MAPTHTT
SCHEMBL7819 0.73 LDHA (0.68) LDHADAOALDH1A1MCL1MEN1
SCHEMBL7300 0.73 LDHA (1.00) LDHADAOALDH1A1MCL1
SCHEMBL7814 0.73 LDHA (1.00) LDHADAOALDH1A1MCL1
SCHEMBL3853249 0.72 MCOLN3 (0.57) KDM4EPKMMCOLN3MAPTHTT
SCHEMBL14118475 0.72 LDHA (0.46) LDHADAOKDM4EHTTPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499114-A1 COMPOUNDS INHIBITORS OF ENZYME LACTATE DEHYDROGENASE (LDH) AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS Universita Di Pisa (IT) 2012-09-19 EP disclosed
WO-2011054525-A1 COMPOUNDS INHIBITORS OF ENZYME LACTATE DEHYDROGENASE (LDH) AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS UNIVERSITA' DI PISA (IT) 2011-05-12 WO disclosed