SCHEMBL1131929

SCHEMBL1131929

COC(=O)/C=C/c1cn(C2CCCCC2)c(-c2ccc(OCc3cc(OC)ccc3-c3ccc(Cl)cc3)cc2)n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 5/20 0.40
CNR1 P21554 4/20 0.37
CNR2 P34972 2/20 0.37
FFAR1 O14842 1/20 0.37
FFAR4 Q5NUL3 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PTGER4 P35408 1/20 0.35
BRD4 O60885 3/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KCNA3 P22001 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1131931 1.00 NR1H4 (0.40) NR1H4CNR1CNR2FFAR1FFAR4
SCHEMBL1131302 0.93 FFAR1 (0.39) NR1H4CNR1CNR2FFAR1FFAR4
SCHEMBL1131301 0.93 FFAR1 (0.39) NR1H4CNR1CNR2FFAR1FFAR4
SCHEMBL1131288 0.86 FFAR1 (0.39) NR1H4CNR1CNR2FFAR1FFAR4
SCHEMBL1131291 0.86 FFAR1 (0.39) NR1H4CNR1CNR2FFAR1FFAR4
SCHEMBL1132049 0.85 PTPN11 (0.37) NR1H4CNR1CNR2FFAR1FFAR4
SCHEMBL1131724 0.85 PTPN11 (0.37) NR1H4CNR1CNR2FFAR1FFAR4
SCHEMBL1131312 0.84 CMKLR1 (0.38) NR1H4CNR1CNR2FFAR1FFAR4
SCHEMBL1131311 0.84 CMKLR1 (0.38) NR1H4CNR1CNR2FFAR1FFAR4
SCHEMBL1131560 0.81 ALOX5 (0.43) NR1H4KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663105-B1 CYCLOALKYL HETEROCYCLES FOR TREATING HEPATITIS C VIRUS BRISTOL MYERS SQUIBB CO (US) 2011-02-16 EP claimed
EP-1663105-B1 CYCLOALKYL HETEROCYCLES FOR TREATING HEPATITIS C VIRUS BRISTOL MYERS SQUIBB CO (US) 2011-02-16 EP disclosed
EP-1663105-B1 CYCLOALKYL HETEROCYCLES FOR TREATING HEPATITIS C VIRUS BRISTOL MYERS SQUIBB CO (US) 2011-02-16 EP disclosed