Pramipexole

Pramipexole

SCHEMBL1132425

CCCN[C@H]1CCc2nc(N)sc2C1.O

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2DRD3DRD4

The experimentally established mechanism targets of Pramipexole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 known ✓ P35462 5/20 0.97
DRD2 known ✓ P14416 5/20 0.97
DRD4 known ✓ P21917 2/20 0.97
HRH2 P25021 2/20 0.97
ADRA2A P08913 2/20 0.97
ADRB2 P07550 1/20 0.97
HTR1A P08908 1/20 0.97
ADRA2B P18089 1/20 0.97
ADRA2C P18825 1/20 0.97
HTR1B P28222 1/20 0.97
HTR2A P28223 1/20 0.97
HTR7 P34969 1/20 0.97
ADRA1A P35348 1/20 0.97
HRH1 P35367 1/20 0.97
HTR2B P41595 1/20 0.97
SIGMAR1 Q99720 1/20 0.97
HRH4 Q9H3N8 1/20 0.97
SCN3A Q9NY46 5/20 0.55
SCN4A P35499 4/20 0.55
SCN9A Q15858 4/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pramipexole SCHEMBL3102892 1.00 DRD3 (0.97) DRD3DRD2DRD4HRH2ADRA2A
Pramipexole SCHEMBL20524815 1.00 DRD3 (0.97) DRD3DRD2DRD4HRH2ADRA2A
Pramipexole SCHEMBL28361114 0.99 DRD3 (1.00) DRD3DRD2DRD4HRH2ADRA2A
Pramipexole SCHEMBL22165339 0.99 DRD3 (1.00) DRD3DRD2DRD4HRH2ADRA2A
Pramipexole SCHEMBL28506481 0.99 DRD3 (1.00) DRD3DRD2DRD4HRH2ADRA2A
Pramipexole SCHEMBL2048695 0.99 DRD3 (1.00) DRD3DRD2DRD4HRH2ADRA2A
Pramipexole SCHEMBL743891 0.99 DRD3 (1.00) DRD3DRD2DRD4HRH2ADRA2A
Dexpramipexole SCHEMBL2289178 0.99 DRD3 (1.00) DRD3DRD2DRD4HRH2ADRA2A
Pramipexole SCHEMBL153875 0.99 DRD3 (1.00) DRD3DRD2DRD4HRH2ADRA2A
Pramipexole SCHEMBL28345162 0.99 DRD3 (1.00) DRD3DRD2DRD4HRH2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2776131-B1 COMPOSITION FOR TREATING OR PREVENTING NEURODEGENERATIVE DISORDERS BIOLOGISCHE HEILMITTEL HEEL GMBH (DE) 2024-05-15 EP claimed
CN-113292440-A Preparation method of N, N-diisopropylethylenediamine and preparation method of pramiperacetam monohydrate 浙江朗华制药有限公司 2021-08-24 CN claimed
CN-113185442-A Pramipexole hydrate crystal and preparation method thereof 许昌远志生物科技有限公司 2021-07-30 CN claimed
CN-111875530-A Pramipexole hydrate crystal and preparation method thereof 浙江朗华制药有限公司 2020-11-03 CN claimed
EP-2870961-B1 Effervescent formulations of pramipexole SANOVEL ILAC SANAYI VE TICARET AS (TR) 2018-07-18 EP claimed
EP-2568999-B1 ACTH FOR TREATMENT OF AMYOTROPHIC LATERAL SCLEROSIS MALLINCKRODT ARD IP LTD (IE) 2018-07-11 EP claimed
EP-2364694-B1 Controlled-release formulations of pramipexole SANOVEL ILAC SANAYI VE TICARET ANONIM SIRKETI (TR) 2013-11-06 EP claimed
EP-1536792-B1 PRAMIPEXOLE ONCE-DAILY DOSAGE FORM PHARMACIA LLC (US) 2013-09-18 EP claimed
EP-2295040-B1 Pharmaceutical compositions of pramipexole SANOVEL ILAC SANAYI VE TICARET AS (TR) 2011-10-12 EP claimed
EP-1781260-B9 EXTENDED RELEASE TABLET FORMULATION CONTAINING PRAMIPEXOLE OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, METHOD FOR MANUFACTURING THE SAME AND USE THEREOF BOEHRINGER INGELHEIM INT (DE) 2011-02-16 EP claimed
EP-1781260-B1 EXTENDED RELEASE TABLET FORMULATION CONTAINING PRAMIPEXOLE OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, METHOD FOR MANUFACTURING THE SAME AND USE THEREOF BOEHRINGER INGELHEIM INT (DE) 2010-11-03 EP claimed
EP-1531814-B1 SUSTAINED-RELEASE TABLET COMPOSITION OF PRAMIPEXOLE PHARMACIA CORP (US) 2008-08-27 EP claimed
US-20240238295-A1 METHOD FOR MODULATING NEUROPATHIES CHENGDU WENDING TECHNOLOGY DEVELOPMENT CO., LTD (CN) 2024-07-18 US disclosed
CN-118056566-A Method and pharmaceutical composition for regulating neuropathy 成都文鼎科技发展有限公司 2024-05-21 CN disclosed
EP-4342471-A1 METHOD FOR MODULATING NEUROPATHIES Chengdu Wending Technology Development Co., Ltd. (CN) 2024-03-27 EP disclosed
CN-117752663-A A method for regulating neuropathy 成都文鼎科技发展有限公司 2024-03-26 CN disclosed
EP-2086536-A1 THE USE OF PRAMIPEXOLE OR A SALT THEREOF FOR THE TREATMENT OF PARKINSON'S DISEASE Boehringer Ingelheim International GmbH (DE) 2009-08-12 EP disclosed
WO-2008104847-A3 PROCESSES FOR THE PREPARATION OF PRAMIPEXOLE AND SALTS THEREOF WOCKHARDT RESEARCH CENTER (IN) 2009-02-05 WO disclosed
WO-2008104847-A2 PROCESSES FOR THE PREPARATION OF PRAMIPEXOLE AND SALTS THEREOF WOCKHARDT RESEARCH CENTRE (IN) 2008-09-04 WO disclosed
WO-2008052953-A1 THE USE OF PRAMIPEXOLE OR A SALT THEREOF FOR THE TREATMENT OF PARKINSON'S DISEASE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-05-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240238295-A1 METHOD FOR MODULATING NEUROPATHIES MME, PMP22, NEFM DRD3 1092/4885DRD2 773/4885DRD4 427/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.