Pramipexole

Pramipexole

SCHEMBL28345162

CCCN[C@H]1CCc2nc(N)sc2C1.Cl.Cl.O.O.O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2DRD3DRD4

The experimentally established mechanism targets of Pramipexole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 known ✓ P35462 5/20 1.00
DRD2 known ✓ P14416 5/20 1.00
DRD4 known ✓ P21917 2/20 1.00
ADRA2A P08913 2/20 0.97
HRH2 P25021 2/20 0.95
ADRB2 P07550 1/20 0.95
HTR1A P08908 1/20 0.95
ADRA2B P18089 1/20 0.95
ADRA2C P18825 1/20 0.95
HTR1B P28222 1/20 0.95
HTR2A P28223 1/20 0.95
HTR7 P34969 1/20 0.95
ADRA1A P35348 1/20 0.95
HRH1 P35367 1/20 0.95
HTR2B P41595 1/20 0.95
SIGMAR1 Q99720 1/20 0.95
HRH4 Q9H3N8 1/20 0.95
SCN3A Q9NY46 5/20 0.54
SCN4A P35499 4/20 0.54
SCN9A Q15858 4/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pramipexole SCHEMBL22165339 1.00 DRD3 (1.00) DRD3DRD2DRD4ADRA2AHRH2
Pramipexole SCHEMBL28361114 1.00 DRD3 (1.00) DRD3DRD2DRD4ADRA2AHRH2
Pramipexole SCHEMBL3947282 1.00 DRD3 (1.00) DRD3DRD2DRD4ADRA2AHRH2
Pramipexole SCHEMBL2048695 1.00 DRD3 (1.00) DRD3DRD2DRD4ADRA2AHRH2
Pramipexole SCHEMBL153875 1.00 DRD3 (1.00) DRD3DRD2DRD4ADRA2AHRH2
Pramipexole SCHEMBL743891 1.00 DRD3 (1.00) DRD3DRD2DRD4ADRA2AHRH2
Dexpramipexole SCHEMBL2289178 1.00 DRD3 (1.00) DRD3DRD2DRD4ADRA2AHRH2
Pramipexole SCHEMBL28506481 1.00 DRD3 (1.00) DRD3DRD2DRD4ADRA2AHRH2
Dexpramipexole SCHEMBL910147 0.99 ADRA2A (1.00) DRD3DRD2DRD4ADRA2AHRH2
Pramipexole SCHEMBL20524815 0.99 DRD3 (0.97) DRD3DRD2DRD4ADRA2AHRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110730662-A NK 1-antagonist combinations and methods for treating synucleinopathies 才思治疗公司 2020-01-24 CN disclosed