SCHEMBL11328530

SCHEMBL11328530

c1ccc2c(c1)CC1CC1c1ccccc1-2

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 8/20 0.50
HTR2C P28335 6/20 0.38
HTR2B P41595 6/20 0.38
HRH3 Q9Y5N1 5/20 0.38
ACHE P22303 2/20 0.37
NOS3 P29474 3/20 0.37
NOS2 P35228 3/20 0.37
TSHR P16473 1/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
CDK8 P49336 1/20 0.34
CDK5 Q00535 1/20 0.34
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29723594 0.83 HTR2A (0.50) HTR2AHTR2CHTR2BHRH3SIGMAR1
SCHEMBL2766554 0.83 HTR2A (0.50) HTR2AHTR2CHTR2BHRH3SIGMAR1
Ammonia Solution, Strong SCHEMBL2786789 0.81 HTR2A (0.49) HTR2AHTR2CHTR2BHRH3SIGMAR1
Hydrochloric Acid SCHEMBL8521423 0.79 HTR2A (0.50) HTR2AHTR2CHTR2BHRH3SIGMAR1
Bromide SCHEMBL7360884 0.79 HTR2A (0.47) HTR2AHTR2CHTR2BHRH3SIGMAR1
Hydrochloric Acid SCHEMBL7424402 0.79 HTR2A (0.50) HTR2AHTR2CHTR2BHRH3SIGMAR1
SCHEMBL13391138 0.76 ACHE (0.56) HTR2AHTR2CHTR2BACHETSHR
SCHEMBL11605889 0.74 HTR2A (0.42) HTR2AHTR2CHTR2BHRH3NOS3
SCHEMBL11328523 0.73 HTR1A (0.43) HTR2AHTR2CHTR2BACHENOS3
SCHEMBL14870745 0.72 HTR2A (0.55) HTR2AACHENOS3NOS2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4258211-A 4-Aminoaliphatic-2,3,5,6-[dibenzobicyclo[5.1.0]octanes] and salts thereof MERCK & CO., INC. (US) 1981-03-24 US disclosed
US-4082801-A 4-Aminomethyldibenzobicyclo[5.1.0]octanes MERCK & CO., INC. (US) 1978-04-04 US disclosed
US-4062891-A N-formyl-2,3,5,6-dibenzobicyclo[5.1.0]octan-4-methylamine MERCK & CO., INC. (US) 1977-12-13 US disclosed
US-3960974-A 4-Halo-2,3,5,6-dibenzobicyclo[5.1.0]octane MERCK & CO., INC. (US) 1976-06-01 US disclosed