SCHEMBL11328751

SCHEMBL11328751

COc1c(Cl)ccc2c1CNCCC2

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.64
ADRA2A P08913 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
HTR2A P28223 4/20 0.42
HTR2C P28335 4/20 0.42
HTR2B P41595 4/20 0.42
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
S1PR1 P21453 1/20 0.38
ADRA1A P35348 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23260194 0.80 PNMT (0.40) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL11327857 0.79 PNMT (0.70) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL476330 0.78 PNMT (1.00) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL30249887 0.78 PNMT (1.00) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL11322725 0.78 HTR2C (0.65) PNMTADRA2AADRA2BADRA2CHTR2A
Hydrochloric Acid SCHEMBL158709 0.77 PNMT (0.96) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL11335328 0.76 PNMT (0.47) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL11340596 0.76 PNMT (0.70) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL11322190 0.76 PNMT (0.70) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL5022472 0.72 PNMT (0.59) PNMTADRA2AADRA2BADRA2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0002624-B1 2-BENZAZEPINE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITHKLINE BECKMAN CORPORATION (US) 1981-10-14 EP disclosed
EP-0002624-A1 2-Benzazepine compounds, processes for their preparation and pharmaceutical compositions containing them SMITHKLINE BECKMAN CORPORATION (US) 1979-06-27 EP disclosed