SCHEMBL11329934

SCHEMBL11329934

c1cc2oc3c(c2cc1C1CCNCC1)CCCC3

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
QDPR P09417 1/20 0.43
TBK1 Q9UHD2 1/20 0.42
TP53 P04637 4/20 0.40
MAPT P10636 4/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
HTR2C P28335 4/20 0.39
HTR6 P50406 2/20 0.38
KMT2A Q03164 1/20 0.38
MAOA P21397 1/20 0.38
SLC18A3 Q16572 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
TLR9 Q9NR96 1/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
NPC1 O15118 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11337723 0.99 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C19QDPRTBK1
SCHEMBL11334573 0.81 CYP1A2 (0.49) CYP1A2CYP3A4CYP2C19QDPRTP53
SCHEMBL11334570 0.78 CYP1A2 (0.49) CYP1A2CYP3A4CYP2C19TP53MAPT
SCHEMBL11338664 0.78 IKBKE (0.48) CYP1A2CYP3A4CYP2C19TBK1TP53
SCHEMBL11332265 0.77 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C19TP53MAPT
SCHEMBL11336420 0.77 CYP1A2 (0.45) CYP1A2CYP3A4CYP2C19TP53MAPT
SCHEMBL11335477 0.76 TSHR (0.43) TP53MAPTBCHEACHEHTR2C
SCHEMBL11334553 0.75 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19TP53MAPT
SCHEMBL11348751 0.74 ACHE (0.51) CYP1A2CYP3A4CYP2C19MAPTBCHE
SCHEMBL11334556 0.74 HTR2C (0.47) QDPRTBK1HTR2CSLC18A3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4259338-A Benzofuranyl-tetrahydropyridines and -piperidines, their acid addition salts and antidepressant preparations thereof CIBA-GEIGY CORPORATION (US) 1981-03-31 US claimed
EP-0006524-A1 Tetrahydropyridine and tetrahydropiperidine derivatives, their acid addition salts, processes for their preparation and pharmaceutical compositions containing them CIBA-GEIGY AG (CH) 1980-01-09 EP claimed
US-4259338-A Benzofuranyl-tetrahydropyridines and -piperidines, their acid addition salts and antidepressant preparations thereof CIBA-GEIGY CORPORATION (US) 1981-03-31 US disclosed
EP-0006524-A1 Tetrahydropyridine and tetrahydropiperidine derivatives, their acid addition salts, processes for their preparation and pharmaceutical compositions containing them CIBA-GEIGY AG (CH) 1980-01-09 EP disclosed