SCHEMBL11337352

SCHEMBL11337352

O=C(O)CCc1ccccc1N1C(=O)c2ccccc2C1=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 4/20 0.67
NR1H2 P55055 3/20 0.67
PPARA Q07869 2/20 0.57
PPARD Q03181 1/20 0.57
PTGER1 P34995 2/20 0.49
PTGER4 P35408 2/20 0.49
PTGER3 P43115 2/20 0.49
PTGER2 P43116 2/20 0.49
CA12 O43570 2/20 0.46
CA9 Q16790 2/20 0.46
ALDH1A1 P00352 3/20 0.45
CYP3A4 P08684 2/20 0.45
HPGD P15428 2/20 0.45
POLB P06746 2/20 0.45
KDM4E B2RXH2 1/20 0.45
TP53 P04637 1/20 0.45
GLA P06280 1/20 0.45
CYP2D6 P10635 1/20 0.45
ALOX12 P18054 1/20 0.45
NFKB1 P19838 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5717701 0.91 NR1H3 (0.63) NR1H3NR1H2PPARAPPARDPTGER1
SCHEMBL28721510 0.86 PTGER4 (0.52) NR1H3NR1H2PPARAPPARDPTGER1
SCHEMBL6690679 0.83 NR1H3 (0.61) NR1H3NR1H2PPARAPPARDCA12
SCHEMBL1904159 0.81 NR1H3 (0.68) NR1H3NR1H2ALDH1A1POLB
SCHEMBL5717824 0.81 NR1H3 (0.62) NR1H3NR1H2PPARAPPARDALDH1A1
SCHEMBL29616419 0.80 NR1H3 (1.00) NR1H3NR1H2PPARAPPARDALDH1A1
SCHEMBL2464969 0.80 NR1H3 (1.00) NR1H3NR1H2PPARAPPARDALDH1A1
SCHEMBL8097081 0.77 CA12 (0.54) PPARAPPARDPTGER1PTGER4PTGER3
SCHEMBL27586782 0.77 NR1H3 (0.70) NR1H3NR1H2POLB
SCHEMBL71453 0.77 PTGER4 (0.68) PTGER1PTGER4PTGER3PTGER2APEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4275217-A Process for the preparation of optically active α-amino acids and their derivatives AGENCE NATIONALE DE VALORISATION DE LA RECHERCHE (ANVAR) (FR) 1981-06-23 US claimed
US-10974235-B2 Targeted, metal-catalyzed fluorination of complex compounds with fluoride ion via decarboxylation TRUSTEES OF PRINCETON UNIVERSITY (US) 2021-04-13 US disclosed
US-20200108380-A1 TARGETED, METAL-CATALYZED FLUORINATION OF COMPLEX COMPOUNDS WITH FLUORIDE ION VIA DECARBOXYLATION THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2020-04-09 US disclosed
US-10543481-B2 Targeted, metal-catalyzed fluorination of complex compounds with fluoride ion via decarboxylation TRUSTEES OF PRINCETON UNIVESITY (US) 2020-01-28 US disclosed
US-20180037526-A1 TARGETED, METAL-CATALYZED FLUORINATION OF COMPLEX COMPOUNDS WITH FLUORIDE ION VIA DECARBOXYLATION THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2018-02-08 US disclosed
WO-2016130549-A1 TARGETED, METAL-CATALYZED FLUORINATION OF COMPLEX COMPOUNDS WITH FLUORIDE ION VIA DECARBOXYLATION THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2016-08-18 WO disclosed
US-20160158388-A1 TARGETED, METAL-CATALYZED FLUORINATION OF COMPLEX COMPOUNDS WITH FLUORIDE ION VIA DECARBOXYLATION THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2016-06-09 US disclosed
US-4275217-A Process for the preparation of optically active α-amino acids and their derivatives AGENCE NATIONALE DE VALORISATION DE LA RECHERCHE (ANVAR) (FR) 1981-06-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160158388-A1 TARGETED, METAL-CATALYZED FLUORINATION OF COMPLEX COMPOUNDS WITH FLUORIDE ION VIA DECARBOXYLATION AFF2, CLTC, AFF4 NR1H3 3254/4885NR1H2 3528/4885PPARA 1655/4885
US-10543481-B2 Targeted, metal-catalyzed fluorination of complex compounds with fluoride ion via decarboxylation AFF2, CLTC, AFF4 NR1H3 3254/4885NR1H2 3528/4885PPARA 1655/4885
US-20180037526-A1 TARGETED, METAL-CATALYZED FLUORINATION OF COMPLEX COMPOUNDS WITH FLUORIDE ION VIA DECARBOXYLATION AFF2, CLTC, AFF4 NR1H3 3254/4885NR1H2 3528/4885PPARA 1655/4885
US-10974235-B2 Targeted, metal-catalyzed fluorination of complex compounds with fluoride ion via decarboxylation AFF2, CLTC, AFF4 NR1H3 3254/4885NR1H2 3528/4885PPARA 1655/4885
US-20200108380-A1 TARGETED, METAL-CATALYZED FLUORINATION OF COMPLEX COMPOUNDS WITH FLUORIDE ION VIA DECARBOXYLATION AFF2, CLTC, AFF4 NR1H3 3254/4885NR1H2 3528/4885PPARA 1655/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.