Ethylenediamine

Ethylenediamine

SCHEMBL11340271

Cc1ccccc1S(=O)(=O)O.NCCN

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3PDE3APDE3BPDE4APDE4BPDE4CPDE4D

The experimentally established mechanism targets of Ethylenediamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.46
RAPGEF4 Q8WZA2 1/20 0.44
SUMO2 P61956 1/20 0.42
SUMO1 P63165 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP3 Q9H4L4 1/20 0.42
SENP2 Q9HC62 1/20 0.42
SENP1 Q9P0U3 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41
CYP1A2 P05177 1/20 0.41
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
CA9 Q16790 3/20 0.40
TTR P02766 1/20 0.40
KMT2A Q03164 2/20 0.40
KAT6A Q92794 1/20 0.40
GAA P10253 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Monoethanolamine SCHEMBL8423206 0.92 MYC (0.43) MYCRAPGEF4SUMO2SUMO1SENP7
Ethylamine SCHEMBL7984887 0.92 RAPGEF4 (0.47) MYCRAPGEF4SUMO2SUMO1SENP7
Hydroxyamine SCHEMBL8185329 0.90 MYC (0.50) MYCRAPGEF4SUMO2SUMO1SENP7
Hydrazine SCHEMBL27884457 0.90 MYC (0.50) MYCRAPGEF4SUMO2SUMO1SENP7
SCHEMBL1748 0.89 MYC (0.53) MYCRAPGEF4SUMO2SUMO1SENP7
SCHEMBL29392580 0.89 MYC (0.53) MYCRAPGEF4SUMO2SUMO1SENP7
Butylamine SCHEMBL6670622 0.88 ALDH1A1 (0.44) MYCRAPGEF4SUMO2SUMO1SENP7
SCHEMBL1557256 0.88 SUMO2 (0.40) MYCRAPGEF4SUMO2SUMO1SENP7
SCHEMBL10492882 0.88 MYC (0.48) MYCRAPGEF4SUMO2SUMO1SENP7
Water SCHEMBL8126703 0.87 MYC (0.52) MYCRAPGEF4SUMO2SUMO1SENP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4254133-A MITICIDE CIBA-GEIGY CORPORATION (US) 1981-03-03 US disclosed
US-4018765-A HETEROCYCLIC HOFFMANN-LA ROCHE INC. (US) 1977-04-19 US disclosed
US-3931217-A ANALGESIC, PSYCHOSTIMULANT HOFFMANN-LA ROCHE INC. (US) 1976-01-06 US disclosed