SCHEMBL11340758

SCHEMBL11340758

NCC(=O)c1ccc(NC(=O)c2ccccc2)c(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.58
KDM4E B2RXH2 2/20 0.58
RXFP1 Q9HBX9 1/20 0.58
MAPT P10636 4/20 0.55
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
SMN1; SMN2 Q16637 2/20 0.54
HSD17B10 Q99714 1/20 0.54
HDAC1 Q13547 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
ALDH1A1 P00352 2/20 0.52
GRM4 Q14833 1/20 0.52
RAB9A P51151 3/20 0.50
LMNA P02545 1/20 0.50
POLB P06746 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
SERPINE1 P05121 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3529060 0.80 MAPT (0.82) NPSR1KDM4ERXFP1MAPTMEN1
SCHEMBL8804658 0.79 KDM4E (0.82) NPSR1KDM4ERXFP1MAPTMEN1
SCHEMBL9362200 0.78 HDAC1 (0.68) NPSR1KDM4ERXFP1MAPTMEN1
SCHEMBL3783679 0.77 GRM4 (0.79) NPSR1KDM4ERXFP1MAPTMEN1
SCHEMBL3528846 0.77 NPSR1 (0.61) NPSR1KDM4ERXFP1MAPTMEN1
SCHEMBL24252964 0.76 MAPT (0.66) NPSR1KDM4ERXFP1MAPTMEN1
SCHEMBL28197181 0.76 RAB9A (0.70) NPSR1KDM4ERXFP1MAPTMEN1
SCHEMBL8980369 0.76 KCNK3 (0.69) MAPTMEN1KMT2ASMN1; SMN2HDAC1
SCHEMBL866785 0.75 MAPT (0.78) NPSR1KDM4ERXFP1MAPTMEN1
SCHEMBL30492552 0.75 MAPT (0.78) NPSR1KDM4ERXFP1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0010030-B1 DERIVATIVES OF 2'-(ORTHO-CHLORO-BENZOYL),4'-CHLORO-GLYCIN ANILIDE, THEIR PREPARATION AND THEIR USE IN MEDICINES PIERRE FABRE S.A. (FR) 1982-05-05 EP claimed
EP-0010030-A1 Derivatives of 2'-(ortho-chloro-benzoyl),4'-chloro-glycin anilide, their preparation and their use in medicines PIERRE FABRE S.A. (FR) 1980-04-16 EP claimed
EP-0044091-A2 Process for the preparation of N-alkylamino-benzophenones PIERRE FABRE S.A. (FR) 1982-01-20 EP disclosed
EP-0010030-A1 Derivatives of 2'-(ortho-chloro-benzoyl),4'-chloro-glycin anilide, their preparation and their use in medicines PIERRE FABRE S.A. (FR) 1980-04-16 EP disclosed