SCHEMBL11344730

SCHEMBL11344730

O=C1CCc2cc(OCCCN3CCN(c4ccc(Cl)cc4)CC3)ccc2N1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.69
DRD2 P14416 11/20 0.66
DRD3 P35462 5/20 0.66
HTR1A P08908 4/20 0.66
HTR2A P28223 4/20 0.66
DRD4 P21917 3/20 0.66
HTR2C P28335 3/20 0.66
SLC6A4 P31645 3/20 0.66
HTR7 P34969 3/20 0.66
MAOA P21397 5/20 0.59
MAOB P27338 4/20 0.59
DRD1 P21728 2/20 0.57
DRD5 P21918 2/20 0.57
HTR3E A5X5Y0 1/20 0.57
MEN1 O00255 1/20 0.57
MLNR O43193 1/20 0.57
HTR3B O95264 1/20 0.57
ABCB11 O95342 1/20 0.57
ESR1 P03372 1/20 0.57
PGR P06401 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10428627 0.93 DRD2 (0.76) KCNH2DRD2DRD3HTR1AHTR2A
SCHEMBL10569598 0.91 KCNH2 (0.66) KCNH2DRD2DRD3HTR1AHTR2A
SCHEMBL23097620 0.91 KCNH2 (0.69) KCNH2DRD2DRD3HTR1AHTR2A
SCHEMBL23097686 0.90 DRD2 (0.64) KCNH2DRD2DRD3HTR1AHTR2A
SCHEMBL23097691 0.90 DRD2 (0.67) KCNH2DRD2DRD3HTR1AHTR2A
SCHEMBL23097641 0.90 DRD2 (0.66) KCNH2DRD2DRD3HTR1AHTR2A
SCHEMBL10571129 0.90 DRD2 (0.68) KCNH2DRD2DRD3HTR1AHTR2A
SCHEMBL10571461 0.90 DRD2 (0.66) KCNH2DRD2DRD3HTR1AHTR2A
SCHEMBL23097597 0.90 DRD2 (0.66) KCNH2DRD2DRD3HTR1AHTR2A
SCHEMBL23097720 0.90 DRD2 (0.75) KCNH2DRD2DRD3HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170334-B1 NMDA RECEPTOR ANTAGONISTS FOR NEUROPROTECTION UNIV EMORY (US) 2021-03-17 EP disclosed
EP-0005828-B1 NEW SUBSTITUTED PHENYLPIPERAZINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION HOECHST AKTIENGESELLSCHAFT (DE) 1981-03-11 EP disclosed