SCHEMBL11348019

SCHEMBL11348019

N#CC1CCn2c(C(=O)c3ccc(F)cc3)ccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.48
RAB9A P51151 4/20 0.48
CDC42 P60953 3/20 0.48
RAC1 P63000 3/20 0.48
PTGS2 P35354 3/20 0.48
PTGS1 P23219 2/20 0.48
CHRM3 P20309 1/20 0.48
OPRM1 P35372 1/20 0.48
PAK1 Q13153 1/20 0.48
LMNA P02545 5/20 0.43
MAPK1 P28482 2/20 0.43
HTT P42858 2/20 0.43
ABCC4 O15439 1/20 0.43
BLM P54132 1/20 0.43
CYP1A2 P05177 1/20 0.43
NFKB1 P19838 1/20 0.43
CTSB P07858 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
CTSC P53634 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11352958 0.87 CDC42 (0.48) NPC1RAB9ACDC42RAC1PTGS2
SCHEMBL11533036 0.87 PTGS2 (0.48) NPC1RAB9ACDC42RAC1PTGS2
SCHEMBL7905025 0.86 PTGS2 (0.64) NPC1RAB9ACDC42RAC1PTGS2
SCHEMBL11350964 0.85 CDC42 (0.47) NPC1RAB9ACDC42RAC1PTGS2
SCHEMBL11346567 0.84 CDC42 (0.45) NPC1RAB9ACDC42RAC1PTGS2
SCHEMBL11442232 0.84 CDC42 (0.45) NPC1RAB9ACDC42RAC1PTGS2
SCHEMBL11444501 0.83 CDC42 (0.44) NPC1RAB9ACDC42RAC1PTGS2
SCHEMBL11442353 0.81 PTGS2 (0.43) NPC1RAB9ACDC42RAC1PTGS2
SCHEMBL11340229 0.81 CDC42 (0.43) NPC1RAB9ACDC42RAC1PTGS2
SCHEMBL11348856 0.81 CDC42 (0.44) NPC1RAB9ACDC42RAC1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000649-B1 5-SUBSTITUTED-1,2-DIHYDRO-3H-PYRROLO(1,2-A)PYRROLE-1-CARBONITRILES AND PROCESS FOR THEIR CONVERSION TO THE CORRESPONDING 1-CARBOXYLIC ACIDS SYNTEX (U.S.A.) INC. (US) 1981-03-25 EP disclosed
US-4140698-A 1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles SYNTEX (USA) INC. (US) 1979-02-20 US disclosed
EP-0000649-A1 5-substituted-1,2-dihydro-3H-pyrrolo(1,2-a)pyrrole-1-carbonitriles and process for their conversion to the corresponding 1-carboxylic acids SYNTEX (U.S.A.) INC. (US) 1979-02-07 EP disclosed