SCHEMBL1135129

SCHEMBL1135129

CCC(/C=C/C(N)=O)N(CC)CC

nearest known ligand 0.30

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GABRP O00591 2/20 0.30
GABRD O14764 2/20 0.30
GABRA1 P14867 2/20 0.30
GABRB1 P18505 2/20 0.30
GABRG2 P18507 2/20 0.30
GABRB3 P28472 2/20 0.30
GABRA5 P31644 2/20 0.30
GABRA3 P34903 2/20 0.30
GABRA2 P47869 2/20 0.30
GABRB2 P47870 2/20 0.30
GABRA4 P48169 2/20 0.30
GABRE P78334 2/20 0.30
GABRA6 Q16445 2/20 0.30
GABRG1 Q8N1C3 2/20 0.30
GABRG3 Q99928 2/20 0.30
GABRQ Q9UN88 2/20 0.30
FDPS P14324 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1486043 1.00 GABRP (0.30) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2773485 0.87
SCHEMBL2384829 0.82 CHRNB2 (0.33)
SCHEMBL2384820 0.82 CHRNB2 (0.33)
SCHEMBL5038530 0.78 GABRP (0.35) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL17183804 0.72 KDM4E (0.39) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL17672256 0.72 CA1 (0.32) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL1135132 0.71 KDM4E (0.30)
SCHEMBL736603 0.71 KDM4E (0.30)
SCHEMBL9607828 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2310104-B1 MIXED GRAFT POLYMERS FOR ION EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2017-10-18 EP claimed
US-8673988-B2 Graft copolymers for ion exchange chromatography MERCK PATENT GMBH (DE) 2014-03-18 US claimed
JP-2011529508-A 2011-12-08 JP claimed
US-20110136925-A1 GRAFT COPOLYMERS FOR ION EXCHANGE CHROMATOGRAPHY MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2011-06-09 US claimed
EP-2310104-A1 GRAFT COPOLYMERS FOR ION EXCHANGE CHROMATOGRAPHY Merck Patent GmbH (DE) 2011-04-20 EP claimed
EP-2153877-A1 Mixed graft polymers for ion exchange chromatography MERCK PATENT GmbH (DE) 2010-02-17 EP claimed
WO-2010012358-A1 GRAFT COPOLYMERS FOR ION EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2010-02-04 WO claimed
US-20220098233-A1 Mixed Bed Ion Exchange Adsorber EMD MILLIPORE CORP (US) 2022-03-31 US disclosed
US-11236125-B2 Mixed bed ion exchange adsorber EMD MILLIPORE CORPORATION (US) 2022-02-01 US disclosed
US-20170298091-A1 Mixed Bed Ion Exchange Adsorber EMD MILLIPORE CORPORATION 2017-10-19 US disclosed
EP-2310104-B1 MIXED GRAFT POLYMERS FOR ION EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2017-10-18 EP disclosed
EP-3230299-A1 MIXED BED ION EXCHANGE ADSORBER EMD Millipore Corporation (US) 2017-10-18 EP disclosed
WO-2016093926-A1 MIXED BED ION EXCHANGE ADSORBER EMD MILLIPORE CORPORATION (US) 2016-06-16 WO disclosed
US-20110136925-A1 GRAFT COPOLYMERS FOR ION EXCHANGE CHROMATOGRAPHY MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2011-06-09 US disclosed
EP-2310104-A1 GRAFT COPOLYMERS FOR ION EXCHANGE CHROMATOGRAPHY Merck Patent GmbH (DE) 2011-04-20 EP disclosed
US-20110073547-A1 Ce(IV)-initiated graft polymerisation on polymers containing no hydroxyl groups MERCK PATENT GESELLSCHAFT (DE) 2011-03-31 US disclosed
EP-2285485-A1 CE(IV)-INITIATED GRAFT POLYMERIZATION ON POLYMERS NOT CONTAINING HYDROXYL GROUPS Merck Patent GmbH (DE) 2011-02-23 EP disclosed
EP-2153877-A1 Mixed graft polymers for ion exchange chromatography MERCK PATENT GmbH (DE) 2010-02-17 EP disclosed
WO-2010012358-A1 GRAFT COPOLYMERS FOR ION EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2010-02-04 WO disclosed
WO-2009143953-A1 CE(IV)-INITIATED GRAFT POLYMERIZATION ON POLYMERS NOT CONTAINING HYDROXYL GROUPS MERCK PATENT GMBH (DE) 2009-12-03 WO disclosed