Nafimidone

Nafimidone

SCHEMBL11356554

C=C.O=C(Cn1ccnc1)c1ccc2ccccc2c1

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPG P10696 2/20 0.63
ALPI P09923 1/20 0.63
TDP1 Q9NUW8 1/20 0.63
PLAA Q9Y263 1/20 0.63
L3MBTL1 Q9Y468 1/20 0.63
CYP19A1 P11511 6/20 0.58
CYP11B1 P15538 2/20 0.57
CYP11B2 P19099 2/20 0.57
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA3 P07451 1/20 0.53
CA4 P22748 1/20 0.53
CA6 P23280 1/20 0.53
CA5A P35218 1/20 0.53
CA7 P43166 1/20 0.53
CA9 Q16790 1/20 0.53
CA13 Q8N1Q1 1/20 0.53
CA14 Q9ULX7 1/20 0.53
CA5B Q9Y2D0 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nafimidone SCHEMBL1817018 0.97 ALPG (0.66) ALPGALPITDP1PLAAL3MBTL1
Nafimidone SCHEMBL29861032 0.96 ALPG (0.67) ALPGALPITDP1PLAAL3MBTL1
Nafimidone SCHEMBL412582 0.96 ALPG (0.67) ALPGALPITDP1PLAAL3MBTL1
Nafimidone SCHEMBL11355091 0.92 ALPG (0.57) ALPGALPITDP1PLAAL3MBTL1
SCHEMBL11481042 0.85 ALPG (0.68) ALPGALPITDP1PLAAL3MBTL1
Ethylene SCHEMBL10973442 0.85 ALPG (0.57) ALPGALPITDP1PLAAL3MBTL1
SCHEMBL11253238 0.84 TBXAS1 (0.56) ALPGALPITDP1PLAAL3MBTL1
Hydrochloric Acid SCHEMBL11181980 0.84 ALPG (0.69) ALPGALPITDP1PLAAL3MBTL1
SCHEMBL11188512 0.84 ALPG (0.63) ALPGALPITDP1PLAAL3MBTL1
SCHEMBL11474959 0.84 ALPG (0.63) ALPGALPITDP1PLAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0001926-B1 1-(NAPHTHYLETHYL)IMIDAZOLE DERIVATIVES, THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SYNTEX (U.S.A.) INC. (US) 1981-04-29 EP disclosed
EP-0001926-A1 1-(Naphthylethyl)imidazole derivatives, their preparation, and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1979-05-16 EP disclosed
US-4150153-A ANTICONVULSANTS, GASTRIC ANTISECRETORY AGENTS SYNTEX (U.S.A.) INC. (US) 1979-04-17 US disclosed