SCHEMBL11366604

SCHEMBL11366604

CCOc1ccc2c(CCBr)c[nH]c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.54
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
HTR6 P50406 1/20 0.51
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
HTR1A P08908 10/20 0.46
HTR1B P28222 8/20 0.46
HTR1D P28221 7/20 0.44
CHRNB2 P17787 1/20 0.43
CHRNA7 P36544 1/20 0.43
CHRNA4 P43681 1/20 0.43
KDM4E B2RXH2 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11362476 0.85 CYP2D6 (0.57) HTR2AMEN1KMT2AHTR6MTNR1A
SCHEMBL2537626 0.85 HTR2A (0.74) HTR2AMEN1KMT2AHTR6HTR1A
SCHEMBL3816723 0.85 HTR2A (0.73) HTR2AMEN1KMT2AHTR6MTNR1A
SCHEMBL11360288 0.81 HTR2A (0.52) HTR2AMEN1KMT2AHTR6MTNR1A
SCHEMBL4604830 0.81 CYP2C19 (0.51) HTR2AMEN1KMT2AHTR6MTNR1A
SCHEMBL4605682 0.79 MTNR1A (0.55) HTR2AMEN1KMT2AHTR6MTNR1A
SCHEMBL27596056 0.79 HTR2A (0.47) HTR2AMEN1KMT2AHTR6MTNR1A
SCHEMBL27596055 0.79 MTNR1A (0.52) HTR2AMEN1KMT2AHTR6MTNR1A
SCHEMBL10919832 0.76 HTR2A (0.71) HTR2AMEN1KMT2AHTR6MTNR1A
SCHEMBL8291070 0.76 ALDH1A1 (0.47) HTR2AMEN1KMT2AHTR6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4255432-A ANTIHYPERTENSIVE AGENTS, ANTIHISTAMINES, BRONCHODILATOR AGENTS, ANTIVASOSPASTIC AGENTS SYNTEX (U.S.A.) INC. (US) 1981-03-10 US disclosed