SCHEMBL11368164

SCHEMBL11368164

COc1ccc(-c2cc3cnccc3c(N)n2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.58
KDM4E B2RXH2 3/20 0.53
GLA P06280 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
DYRK1A Q13627 1/20 0.50
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48
CYP2C19 P33261 1/20 0.48
NPC1 O15118 5/20 0.47
RAB9A P51151 4/20 0.47
CASP3 P42574 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
PRKCH P24723 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11370533 0.89 SYK (0.58) SYKKDM4EGLANPSR1RXFP1
SCHEMBL11373416 0.85 KDM4E (0.58) SYKKDM4EGLANPSR1RXFP1
SCHEMBL11374306 0.83 PRKCD (0.56) CYP1A2PRKCHPRKCEPRKCQPRKCD
SCHEMBL31375795 0.83 PRKCD (0.56) CYP1A2PRKCHPRKCEPRKCQPRKCD
SCHEMBL11366860 0.81 PRKCD (0.45) KDM4ECYP1A2RAB9APRKCHPRKCE
SCHEMBL11375277 0.80 KDM4E (0.50) KDM4EGLACYP1A2CYP3A4CYP2D6
SCHEMBL508360 0.78 SYK (0.56) SYKKDM4EDYRK1ANPC1RAB9A
SCHEMBL11366250 0.78 CYP1A2 (0.51) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11365506 0.77 LATS1 (0.47) CYP1A2PRKCHPRKCEPRKCQPRKCD
SCHEMBL11365490 0.77 ALDH1A1 (0.47) NPSR1DYRK1ACYP2D6CYP2C9CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4260759-A CONDENSATION OF NITRILES SCHERING-CORPORATION (US) 1981-04-07 US disclosed
US-4115395-A FUNGICIDES, BACTERICIDES SCHERING CORPORATION (US) 1978-09-19 US disclosed
US-4107166-A ANTIFUNGAL, ANTIBACTERIAL SCHERING CORPORATION (US) 1978-08-15 US disclosed
US-4017500-A FUNGICIDES, BACTERICIDES SCHERING CORPORATION (US) 1977-04-12 US disclosed