SCHEMBL11370533

SCHEMBL11370533

COc1ccc(-c2cc3ccncc3c(N)n2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.58
KDM4E B2RXH2 3/20 0.53
GLA P06280 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
DYRK1A Q13627 1/20 0.50
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48
CYP2C19 P33261 1/20 0.48
NPC1 O15118 5/20 0.47
RAB9A P51151 4/20 0.47
CASP3 P42574 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
IDO1 P14902 2/20 0.46
TDO2 P48775 2/20 0.46
MEN1 O00255 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11368164 0.89 SYK (0.58) SYKKDM4EGLANPSR1RXFP1
SCHEMBL11370578 0.85 KDM4E (0.58) SYKKDM4EGLANPSR1RXFP1
SCHEMBL11373185 0.83 PRKCH (0.47) KDM4ECYP1A2POLBMAPT
SCHEMBL4772977 0.83 NPC1 (0.47) SYKKDM4EGLANPSR1RXFP1
SCHEMBL11373275 0.81 ADORA2A (0.43) KDM4EGLACYP1A2CYP3A4CYP2C9
SCHEMBL6634946 0.80 KDM4E (0.51) KDM4EGLAIDO1TDO2MEN1
SCHEMBL4253191 0.79 KDM4E (0.51) SYKKDM4EGLANPSR1RXFP1
SCHEMBL11371126 0.78 CYP1A2 (0.51) KDM4ECYP1A2CYP11B1CYP11B2NPC1
SCHEMBL509858 0.78 SYK (0.56) SYKKDM4EDYRK1ANPC1RAB9A
SCHEMBL11367176 0.77 KIF11 (0.46) KDM4EIDO1TDO2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4260759-A CONDENSATION OF NITRILES SCHERING-CORPORATION (US) 1981-04-07 US disclosed
US-4115395-A FUNGICIDES, BACTERICIDES SCHERING CORPORATION (US) 1978-09-19 US disclosed
US-4107166-A ANTIFUNGAL, ANTIBACTERIAL SCHERING CORPORATION (US) 1978-08-15 US disclosed
US-4017500-A FUNGICIDES, BACTERICIDES SCHERING CORPORATION (US) 1977-04-12 US disclosed