SCHEMBL11368351

SCHEMBL11368351

O=C(O)CC1NC(=O)c2c(Cl)cccc21

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
HTR2B P41595 2/20 0.47
PBRM1 Q86U86 8/20 0.46
HSD17B10 Q99714 1/20 0.43
CYP1A2 P05177 1/20 0.42
KMT2A Q03164 1/20 0.39
AKR1B1 P15121 1/20 0.39
GAA P10253 1/20 0.38
SMARCA2 P51531 1/20 0.38
SMARCA4 P51532 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11367617 0.82 CYP1A2 (0.66) HTR2AHTR2CHTR2BPBRM1HSD17B10
SCHEMBL11350233 0.82 HSD17B10 (0.43) PBRM1HSD17B10CYP1A2KMT2AGAA
SCHEMBL11352016 0.79 KDM4E (0.47) HSD17B10CYP1A2GAA
SCHEMBL11355710 0.77 HTR2A (0.45) HTR2AHTR2CHTR2BPBRM1CYP1A2
SCHEMBL31133079 0.74 HSD17B10 (0.73) HTR2AHTR2CHTR2BHSD17B10CYP1A2
SCHEMBL18215418 0.74 HSD17B10 (0.73) HTR2AHTR2CHTR2BHSD17B10CYP1A2
SCHEMBL2645035 0.74 HSD17B10 (0.73) HTR2AHTR2CHTR2BHSD17B10CYP1A2
SCHEMBL18215470 0.74 HSD17B10 (0.73) HTR2AHTR2CHTR2BHSD17B10CYP1A2
SCHEMBL11363508 0.73 HSD17B10 (0.47) HSD17B10CYP1A2GAA
SCHEMBL11354534 0.70 CYP1A2 (0.48) HTR2AHTR2CHTR2BPBRM1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4244966-A 1,3-Dihydro-3-(2-hydroxy-, 2-bromo- or 2-chloroethyl)-2H-isoindol-1-one derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1981-01-13 US disclosed