SCHEMBL11352016

SCHEMBL11352016

COc1cccc2c1C(=O)NC2CC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HPGD P15428 2/20 0.47
CYP1A2 P05177 1/20 0.43
POLL Q9UGP5 1/20 0.43
ALDH1A1 P00352 3/20 0.41
CTH P32929 1/20 0.41
TP53 P04637 1/20 0.41
HSD17B10 Q99714 2/20 0.41
POLB P06746 4/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
ATM Q13315 1/20 0.39
CYP3A4 P08684 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11363652 0.87 CYP1A2 (0.48) KDM4ESMN1; SMN2HPGDCYP1A2POLL
SCHEMBL11350233 0.79 HSD17B10 (0.43) KDM4ESMN1; SMN2HPGDCYP1A2HSD17B10
SCHEMBL11368351 0.79 HTR2A (0.47) CYP1A2HSD17B10GAA
SCHEMBL11362493 0.79 POLL (0.42) KDM4EHPGDCYP1A2POLLALDH1A1
SCHEMBL19249656 0.77 POLL (0.51) KDM4EHPGDPOLLALDH1A1TP53
SCHEMBL11367277 0.73 ATM (0.56) KDM4ECYP1A2ALDH1A1HSD17B10CA1
SCHEMBL31133079 0.72 HSD17B10 (0.73) CYP1A2HSD17B10GAA
SCHEMBL18215418 0.72 HSD17B10 (0.73) CYP1A2HSD17B10GAA
SCHEMBL18215470 0.72 HSD17B10 (0.73) CYP1A2HSD17B10GAA
SCHEMBL2645035 0.72 HSD17B10 (0.73) CYP1A2HSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4244966-A 1,3-Dihydro-3-(2-hydroxy-, 2-bromo- or 2-chloroethyl)-2H-isoindol-1-one derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1981-01-13 US disclosed