SCHEMBL11354534

SCHEMBL11354534

CC(=O)CC1NC(=O)c2c(C)cccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.48
HTR2A P28223 4/20 0.47
HTR2C P28335 4/20 0.47
HTR2B P41595 4/20 0.47
HSD17B10 Q99714 1/20 0.47
PBRM1 Q86U86 6/20 0.39
GAA P10253 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C19 P33261 1/20 0.39
TSHR P16473 2/20 0.35
TNKS2 Q9H2K2 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12718314 0.81 HTR2A (0.51) CYP1A2HTR2AHTR2CHTR2BHSD17B10
SCHEMBL11358191 0.78 HTR2A (0.46) CYP1A2HTR2AHTR2CHTR2BHSD17B10
SCHEMBL13995842 0.76 HSD17B10 (0.71) CYP1A2HTR2AHTR2CHTR2BHSD17B10
SCHEMBL11358726 0.74 HTR2A (0.54) CYP1A2HTR2AHTR2CHTR2BPBRM1
SCHEMBL12716352 0.72 HTR2A (0.55) CYP1A2HTR2AHTR2CHTR2BPBRM1
SCHEMBL29010215 0.71 HTR2A (0.51) CYP1A2HTR2AHTR2CHTR2BPBRM1
SCHEMBL3748724 0.71 HTR2A (0.48) CYP1A2HTR2AHTR2CHTR2BHSD17B10
SCHEMBL11352016 0.71 KDM4E (0.47) CYP1A2HSD17B10GAAALDH1A1HPGD
SCHEMBL11367617 0.71 CYP1A2 (0.66) CYP1A2HTR2AHTR2CHTR2BHSD17B10
SCHEMBL11363644 0.71 CYP1A2 (0.66) CYP1A2HSD17B10PBRM1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4244966-A 1,3-Dihydro-3-(2-hydroxy-, 2-bromo- or 2-chloroethyl)-2H-isoindol-1-one derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1981-01-13 US disclosed