SCHEMBL11368783

SCHEMBL11368783

COc1cccc(C(=O)NC[Sn])c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.64
NPC1 O15118 4/20 0.62
RAB9A P51151 4/20 0.62
HPGD P15428 3/20 0.62
GAA P10253 2/20 0.62
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
ALDH1A1 P00352 1/20 0.59
MAPT P10636 1/20 0.59
SMN1; SMN2 Q16637 3/20 0.59
CES2 O00748 1/20 0.59
CES1 P23141 1/20 0.59
TDP1 Q9NUW8 1/20 0.58
TSHR P16473 2/20 0.57
NPSR1 Q6W5P4 1/20 0.57
TAS1R3 Q7RTX0 1/20 0.57
TAS1R1 Q7RTX1 1/20 0.57
LMNA P02545 1/20 0.57
RXFP1 Q9HBX9 1/20 0.56
KCNK3 O14649 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL47353 0.85 MMP13 (0.66) MMP13NPC1RAB9AHPGDGAA
SCHEMBL11246936 0.84 MMP13 (0.64) MMP13NPC1RAB9AHPGDGAA
SCHEMBL11354985 0.83 KDM4E (0.67) NPC1RAB9AHPGDGAAMEN1
SCHEMBL31178805 0.83 MAPK1 (0.72) MMP13NPC1RAB9AHPGDGAA
SCHEMBL8947214 0.83 MAPK1 (0.72) MMP13NPC1RAB9AHPGDGAA
SCHEMBL30098865 0.83 ALDH1A1 (0.73) MMP13NPC1RAB9AHPGDGAA
SCHEMBL11756934 0.83 GAA (0.73) MMP13NPC1RAB9AHPGDGAA
SCHEMBL9491894 0.83 GAA (0.73) MMP13NPC1RAB9AHPGDGAA
SCHEMBL5672356 0.83 HPGD (0.72) MMP13NPC1RAB9AHPGDGAA
SCHEMBL6361446 0.83 GAA (0.73) MMP13NPC1RAB9AHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362875-A Process for preparing (1-acylaminomethyl)-1,2,3,4-tetrahydroisoquinolines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1982-12-07 US disclosed