SCHEMBL11375868

SCHEMBL11375868

CN(C)c1ccc(C2(N(c3ccccc3)c3ccccc3)OC(=O)c3cc(N(C)C)ccc32)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.63
HPGD P15428 5/20 0.63
TDP1 Q9NUW8 4/20 0.63
CYP3A4 P08684 2/20 0.63
HIF1A Q16665 1/20 0.63
HSD17B10 Q99714 1/20 0.63
MEN1 O00255 6/20 0.51
KMT2A Q03164 6/20 0.51
CRHBP P24387 2/20 0.34
CRHR2 Q13324 2/20 0.34
PKM P14618 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 5/20 0.33
MAPK1 P28482 4/20 0.33
RAB9A P51151 4/20 0.33
LMNA P02545 3/20 0.33
APP P05067 2/20 0.33
PDGFRB P09619 2/20 0.33
SNCA P37840 2/20 0.33
NPC1 O15118 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11448925 1.00 ALDH1A1 (0.63) ALDH1A1HPGDTDP1CYP3A4HIF1A
SCHEMBL11374917 0.96 ALDH1A1 (0.68) ALDH1A1HPGDTDP1CYP3A4HIF1A
SCHEMBL11441974 0.89 TDP1 (0.48) ALDH1A1HPGDTDP1CYP3A4HIF1A
SCHEMBL11377272 0.89 TDP1 (0.48) ALDH1A1HPGDTDP1CYP3A4HIF1A
SCHEMBL11380017 0.89 CYP3A4 (0.51) ALDH1A1HPGDTDP1CYP3A4HIF1A
SCHEMBL9617636 0.86 ALDH1A1 (0.61) ALDH1A1HPGDTDP1CYP3A4HIF1A
SCHEMBL11370697 0.86 ALDH1A1 (0.50) ALDH1A1HPGDTDP1CYP3A4HIF1A
SCHEMBL11422435 0.86 ALDH1A1 (0.50) ALDH1A1HPGDTDP1CYP3A4HIF1A
SCHEMBL11456350 0.84 TDP1 (0.50) ALDH1A1HPGDTDP1CYP3A4HIF1A
SCHEMBL11374410 0.83 NPSR1 (0.47) ALDH1A1HPGDTDP1CYP3A4HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4255577-A Process and intermediates for preparing 3-[4-(disubstituted-amino)phenyl] or STERLING DRUG INC. (US) 1981-03-10 US disclosed
US-4200313-A Carbonless duplicating systems STERLING DRUG INC. (US) 1980-04-29 US disclosed
US-4187223-A 3-[4-(Disubstituted-amino)phenyl]-3-(diphenylamino)phthalides STERLING DRUG INC. (US) 1980-02-05 US disclosed
US-4168378-A THERMOGRAPHY, LEUCO DYES STERLING DRUG INC. (US) 1979-09-18 US disclosed